SCHEMBL12417898

SCHEMBL12417898

CS(=O)(=O)c1cc(F)ccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 1/20 0.37
CCR1 P32246 6/20 0.35
KCNH2 Q12809 2/20 0.35
PTGS2 P35354 2/20 0.35
HTR6 P50406 1/20 0.34
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34
CDK9 P50750 1/20 0.34
CCR2 P41597 1/20 0.33
ADRB1 P08588 1/20 0.33
RIPK2 O43353 1/20 0.33
CYP3A4 P08684 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20084399 0.79 ALDH1A1 (0.33) HTR6CCNB2CDK1CCNB1CCNA2
SCHEMBL10920036 0.77 ROCK1 (0.40) PTGS2
SCHEMBL2642775 0.77 SYK (0.32) SCN10APIK3C3SLC22A12
SCHEMBL2643186 0.77 UHRF1 (0.48) CCR1PTGS2
SCHEMBL2643084 0.75 L3MBTL1 (0.42) PIK3C3
SCHEMBL1404011 0.75 SYK (0.33) PTGS2SCN10APIK3C3
SCHEMBL2643081 0.75 SCN10A (0.33) SCN10APIK3C3
SCHEMBL2642777 0.75 SYK (0.31) SCN10APIK3C3
SCHEMBL2643183 0.75 SYK (0.31) PTGS2SCN10APIK3C3
Hydrochloric Acid SCHEMBL18228284 0.73 L3MBTL1 (0.41) PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110172275-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 US disclosed
US-20110172275-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110172275-A1 PYRROLE COMPOUNDS PRLHR, C1R, C1S TGFBR1 3934/4885CCR1 549/4885KCNH2 348/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.