SCHEMBL12423367

SCHEMBL12423367

CCOC(=O)c1c(C(C)C)nc2c(c1C1=CCCC1)C(O)CC(C)(C)C2

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CETP P11597 17/20 0.43
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10196403 1.00 CETP (0.43) CETPLMNAGAAHTTCYP1A2
SCHEMBL663765 0.88 CETP (0.47) CETP
SCHEMBL16359992 0.85 CETP (0.34) CETPLMNAGAAHTTCYP1A2
SCHEMBL10196417 0.85 CETP (0.34) CETPLMNAGAAHTTCYP1A2
SCHEMBL663475 0.83 CYP1A2 (0.52) LMNAGAAHTTCYP1A2CYP2C9
SCHEMBL12423364 0.79 CETP (0.45) CETPLMNAGAAHTTCYP1A2
SCHEMBL10196397 0.79 CETP (0.45) CETPLMNAGAAHTTCYP1A2
SCHEMBL10196449 0.78 CETP (0.40) CETP
SCHEMBL16258486 0.78 CETP (0.40) CETP
SCHEMBL16363068 0.77 CETP (0.41) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536733-B1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INT (DE) 2014-11-26 EP disclosed
WO-2011101424-A1 TRICYCLIC PYRIDINE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR PREPARATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-25 WO disclosed