SCHEMBL1242422

SCHEMBL1242422

Cc1cnc2ccc(N3CC[C@H](c4cc(F)c(F)cc4F)[C@@H](NC(=O)O)C3)nc2n1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.55
DPP7 Q9UHL4 17/20 0.55
DPP8 Q6V1X1 12/20 0.55
DPP9 Q86TI2 12/20 0.55
CYP2D6 P10635 5/20 0.46
KCNH2 Q12809 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12891146 0.83 DPP4 (0.65) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL8262492 0.83 DPP4 (0.65) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL5109946 0.82 DPP4 (0.55) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL1242439 0.80 DPP4 (0.49) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL1241000 0.76 DPP4 (0.47) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL1240995 0.76 DPP4 (0.47) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL1243362 0.75 DPP4 (0.71) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL2937242 0.75 DPP4 (0.48) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL12891125 0.70 DPP4 (0.84) DPP4DPP7DPP8DPP9CYP2D6
SCHEMBL8261933 0.70 DPP4 (0.84) DPP4DPP7DPP8DPP9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884104-B2 Such as (3R,4R)-1-Pyrimidin-4-yl-4-(2,4,5-trifluorophenyl)piperidin-3-amine bis-trifluoroacetic acid salt MERCK SHARP & DOHME CORP. (US) 2011-02-08 US disclosed