SCHEMBL1242439

SCHEMBL1242439

Nc1ccc(N2CC[C@H](c3cc(F)c(F)cc3F)[C@@H](NC(=O)O)C2)nc1N

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.49
DPP9 Q86TI2 14/20 0.49
DPP7 Q9UHL4 13/20 0.49
DPP8 Q6V1X1 12/20 0.49
CYP2D6 P10635 6/20 0.45
KCNH2 Q12809 6/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1240995 0.88 DPP4 (0.47) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL1241000 0.88 DPP4 (0.47) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL1242422 0.80 DPP4 (0.55) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL5116792 0.78 DPP4 (0.50) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL1243362 0.77 DPP4 (0.71) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL2937242 0.77 DPP4 (0.48) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL5123894 0.70 SIGMAR1 (0.51) DPP4
SCHEMBL1240975 0.70 SIGMAR1 (0.51) DPP4
SCHEMBL1240711 0.70 DPP4 (0.47) DPP4DPP9DPP7DPP8CYP2D6
SCHEMBL5924025 0.69 DPP4 (0.37) DPP4DPP9DPP7DPP8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884104-B2 Such as (3R,4R)-1-Pyrimidin-4-yl-4-(2,4,5-trifluorophenyl)piperidin-3-amine bis-trifluoroacetic acid salt MERCK SHARP & DOHME CORP. (US) 2011-02-08 US disclosed