SCHEMBL1243362

SCHEMBL1243362

Cc1nnc2ccc(N3CC[C@H](c4cc(F)c(F)cc4F)[C@@H](NC(=O)O)C3)nn12

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 17/20 0.71
DPP7 Q9UHL4 10/20 0.71
CYP2D6 P10635 5/20 0.71
KCNH2 Q12809 5/20 0.71
DPP9 Q86TI2 9/20 0.56
DPP8 Q6V1X1 8/20 0.56
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL1240926 0.83 DPP4 (1.00) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL8261870 0.82 DPP4 (0.84) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL12891144 0.82 DPP4 (0.84) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL5114076 0.81 DPP4 (0.71) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL1242439 0.77 DPP4 (0.49) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL1242422 0.75 DPP4 (0.55) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL2937242 0.74 DPP4 (0.48) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL1241000 0.73 DPP4 (0.47) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL1240995 0.73 DPP4 (0.47) DPP4DPP7CYP2D6KCNH2DPP9
SCHEMBL8261904 0.69 DPP4 (0.88) DPP4DPP7CYP2D6KCNH2DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884104-B2 Such as (3R,4R)-1-Pyrimidin-4-yl-4-(2,4,5-trifluorophenyl)piperidin-3-amine bis-trifluoroacetic acid salt MERCK SHARP & DOHME CORP. (US) 2011-02-08 US disclosed