SCHEMBL12425623

SCHEMBL12425623

CCOC(=O)N1C2CCC1CN(C(=O)c1ccc(N)nc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.49
RAB9A P51151 1/20 0.48
HDAC1 Q13547 1/20 0.41
GAA P10253 3/20 0.41
KMT2A Q03164 3/20 0.41
HPGD P15428 2/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
CHRM1 P11229 4/20 0.40
SSTR5 P35346 1/20 0.40
MTOR P42345 1/20 0.39
ADRA1A P35348 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2300794 0.85 HDAC1 (0.52) CDK4HDAC1KMT2AMEN1JAK1
SCHEMBL2301926 0.81 HDAC1 (0.48) CDK4HDAC1KMT2AMEN1CHRM1
SCHEMBL29230240 0.80 RAB9A (0.72) RAB9AGAAKMT2AHPGDMEN1
SCHEMBL31697610 0.80 RAB9A (0.72) RAB9AGAAKMT2AHPGDMEN1
SCHEMBL12425424 0.79 HDAC1 (0.49) HDAC1
SCHEMBL2304154 0.78 GABRP (0.45) CDK4HDAC1HPGDMTORADRA1A
SCHEMBL12425364 0.77 HDAC1 (0.52) RAB9AHDAC1KMT2AMEN1NPSR1
SCHEMBL12425269 0.77 CDK4 (0.50) CDK4HDAC1MTORADRA1AGABRP
SCHEMBL12426761 0.75 CDK4 (0.51) CDK4HDAC1HPGDMTORGABRP
SCHEMBL12426731 0.72 CDK1 (0.47) CDK4HDAC1HPGDMTORGABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101409-A1 PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6 NOVARTIS AG (CH) 2011-08-25 WO disclosed