SCHEMBL12428182

SCHEMBL12428182

CCC1CCCN(CCN2CCn3c(c(C4CCCCC4)c4ccc(C(=O)O)cc43)-c3ccc(OCc4ccccc4)cc32)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.42
MMP12 P39900 1/20 0.42
KDM2B Q8NHM5 2/20 0.41
LTA4H P09960 1/20 0.38
EPHX2 P34913 1/20 0.38
NR1I2 O75469 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
EGFR P00533 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NPY1R P25929 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA5 P30532 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12428227 0.94 PRKCA (0.41) PRKCAMMP12KDM2BLTA4HEPHX2
SCHEMBL12428179 0.93 PRKCA (0.41) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12428247 0.92 PRKCA (0.43) PRKCAMMP12KDM2BNR1I2CYP3A4
SCHEMBL13286276 0.91 PRKCA (0.41) PRKCAMMP12KDM2BNR1I2CYP3A4
SCHEMBL10283489 0.91 EGFR (0.44) PRKCAMMP12EGFRKDM4EALDH1A1
SCHEMBL12428353 0.90 PRKCA (0.39) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL10283245 0.88 PRKCA (0.47) PRKCAMMP12KDM2BNR1I2CYP3A4
SCHEMBL12428189 0.88 PRKCA (0.42) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12428298 0.87 PRKCA (0.40) PRKCAMMP12NR1I2CYP3A4CYP2C9
SCHEMBL12429156 0.87 PRKCA (0.40) PRKCAMMP12NR1I2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed
US-7977331-B1 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor JAPAN TOBACCO INC. (JP) 2011-07-12 US disclosed