SCHEMBL12436769

SCHEMBL12436769

CCNC(=O)NC1CCC(C(C)=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 13/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KDM1A O60341 1/20 0.47
MAOB P27338 1/20 0.47
FASN P49327 1/20 0.45
EPHX2 P34913 4/20 0.43
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22722007 1.00 EPHX1 (0.47) EPHX1KDM4EALDH1A1KDM1AMAOB
SCHEMBL965926 0.88
SCHEMBL15263332 0.88 EPHX1 (0.57) EPHX1KDM4EALDH1A1KDM1AMAOB
SCHEMBL1908654 0.85 EPHX1 (0.50) EPHX1KDM4EALDH1A1KDM1AMAOB
SCHEMBL12436784 0.84 EPHX2 (0.56) EPHX1KDM4EALDH1A1EPHX2KMT2A
SCHEMBL22722017 0.84 EPHX2 (0.56) EPHX1KDM4EALDH1A1EPHX2KMT2A
SCHEMBL20233001 0.81 EPHX1 (0.60) EPHX1KDM4EALDH1A1KDM1AMAOB
SCHEMBL12801142 0.81 EPHX2 (0.65) EPHX1KDM4EALDH1A1KDM1AMAOB
SCHEMBL968340 0.80 EPHX1 (0.63) EPHX1KDM4EALDH1A1EPHX2KMT2A
SCHEMBL965080 0.80 EPHX1 (0.69) EPHX1KDM4EALDH1A1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE48334-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-12-01 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed
WO-2010032856-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME 武田薬品工業株式会社 (JP) 2010-03-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME NTSR2, BDKRB1, AVPR1B EPHX1 3088/4885KDM4E 4083/4885ALDH1A1 3648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.