SCHEMBL12437375

SCHEMBL12437375

CC(=O)[C@H]1CC[C@H](NC(=O)c2cccc(F)n2)CC1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRKAA2 P54646 2/20 0.47
HSD11B1 P28845 2/20 0.45
CD38 P28907 2/20 0.45
CNR2 P34972 2/20 0.42
GRM4 Q14833 2/20 0.41
P2RX7 Q99572 1/20 0.40
EPHX2 P34913 1/20 0.40
SMYD3 Q9H7B4 2/20 0.40
PARP1 P09874 1/20 0.39
DPP4 P27487 1/20 0.39
CLK1 P49759 1/20 0.39
CLK2 P49760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12513462 1.00 PRKAA2 (0.47) PRKAA2HSD11B1CD38CNR2GRM4
SCHEMBL19701368 0.83 SMYD3 (0.50) PRKAA2HSD11B1SMYD3
SCHEMBL21489946 0.83 SMYD3 (0.50) PRKAA2HSD11B1SMYD3
SCHEMBL26412830 0.83 HSD11B1 (0.63) PRKAA2HSD11B1CD38CNR2PARP1
SCHEMBL31514789 0.81 CNR2 (0.59) PRKAA2HSD11B1CNR2GRM4
SCHEMBL23575973 0.79 SMYD3 (0.65) SMYD3
SCHEMBL19710214 0.79 SMYD3 (0.65) SMYD3
SCHEMBL22722015 0.78 SMYD3 (0.64) SMYD3
SCHEMBL12436733 0.78 SMYD3 (0.64) SMYD3
SCHEMBL20103216 0.73 HTR1F (0.45) GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-RE48334-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-12-01 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME NTSR2, BDKRB1, AVPR1B PRKAA2 4122/4885HSD11B1 1352/4885CD38 987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.