SCHEMBL12438703

SCHEMBL12438703

CNC(=O)c1cc(Br)cc(C)c1NC(=O)C1CC(Cl)=NN1c1ncccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 13/20 0.41
DHODH Q02127 1/20 0.34
GRM4 Q14833 1/20 0.34
F10 P00742 1/20 0.34
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9290241 0.93 MALT1 (0.41) MALT1DHODHGRM4F10TRPV1
SCHEMBL12574860 0.91 MALT1 (0.42) MALT1DHODHTRPV1
SCHEMBL9290211 0.91 MALT1 (0.44) MALT1GRM4TRPV1
SCHEMBL9289049 0.91 MALT1 (0.40) MALT1DHODHGRM4F10
SCHEMBL12575514 0.90 MALT1 (0.41) MALT1GRM4TRPV1
SCHEMBL9290246 0.89 MALT1 (0.39) MALT1DHODHTRPV1
SCHEMBL9290062 0.88 MALT1 (0.40) MALT1
SCHEMBL1148395 0.86 MALT1 (0.43) MALT1DHODHGRM4
SCHEMBL9290207 0.86 MALT1 (0.40) MALT1TRPV1
SCHEMBL12438369 0.85 MALT1 (0.40) MALT1DHODHGRM4TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012092827-A1 CHEMICAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2012-07-12 WO disclosed
WO-2011095462-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-08-11 WO disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2010135914-A1 NEW SPIROHETEROCYCLIC FURAN AND THIOFURAN DIONE DERIVATIVES SYNGENTA PARTICIPATIONS AG (CH) 2010-12-02 WO disclosed
WO-2010063670-A1 SPIROHETEROCYCLIC N-OXYAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-10 WO disclosed
EP-1919903-B1 BICYCLIC BISAMIDE DERIVATIVES AND USE THEREOF AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-01-27 EP disclosed
WO-2009024341-A2 CONDENSED ANTHRAN I LAMI DE DERIVATIVES AS INSECTISIDES SYNGENTA PARTICIPATIONS AG, (CH) 2009-02-26 WO disclosed
WO-2009021717-A2 PESTICIDAL FORMULATION SYNGENTA PARTICIPATIONS AG (CH) 2009-02-19 WO disclosed
WO-2009010260-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-01-22 WO disclosed
EP-1819695-B1 ANTHRANILAMIDE DERIVATIVES AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-12-17 EP disclosed
WO-2008064891-A1 N-CYANOALKYLANTHRANILAMIDES AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-06-05 WO disclosed