SCHEMBL12440388

SCHEMBL12440388

Cc1nc2cc3c(cc2[nH]1)CCOCC3

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
MAPT P10636 5/20 0.42
KDM4E B2RXH2 5/20 0.42
POLB P06746 5/20 0.42
HPGD P15428 5/20 0.42
ALDH1A1 P00352 6/20 0.42
HSP90AA1 P07900 1/20 0.38
ESR2 Q92731 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GAA P10253 2/20 0.37
HSD17B10 Q99714 2/20 0.37
RAB9A P51151 6/20 0.36
NPC1 O15118 5/20 0.36
SMN1; SMN2 Q16637 5/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PKM P14618 1/20 0.36
HCRTR1 O43613 1/20 0.35
NFKB1 P19838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12438622 0.92 CHRNB2 (0.40) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL3478940 0.84 CHRNB2 (0.46) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL13998791 0.84 CHRNB2 (0.46) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL12440387 0.83 CHRNB2 (0.38) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL12438640 0.82 CHRNB2 (0.45) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL14648511 0.82 CHRNB2 (0.45) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL720947 0.81 CHRNB2 (0.47) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL12966011 0.81 CHRNB2 (0.40) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL12438620 0.80 CHRNB2 (0.41) CHRNB2CHRNA4MAPTKDM4EPOLB
SCHEMBL719765 0.79 DRD2 (0.44) CHRNB2CHRNA4MAPTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2532665-B1 BENZIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS AND USES THEREOF XUANZHU PHARMA CO LTD (CN) 2016-09-07 EP disclosed
EP-2532665-A1 BENZIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS AND USES THEREOF Xuanzhu Pharma Co., Ltd. (CN) 2012-12-12 EP disclosed
WO-2011095057-A1 BENZIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS AND USES THEREOF 山东轩竹医药科技有限公司 (CN) 2011-08-11 WO disclosed