SCHEMBL12440446

SCHEMBL12440446

Clc1ccc(-c2ccc(-c3cccc(OCCCN4CCCC4)c3)nc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.56
MCHR1 Q99705 4/20 0.54
LTA4H P09960 1/20 0.54
BACE1 P56817 1/20 0.53
HRH1 P35367 1/20 0.52
KCNH2 Q12809 1/20 0.52
CYP2D6 P10635 1/20 0.51
CHRM1 P11229 1/20 0.51
HTR2A P28223 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12439987 0.94 LTA4H (0.62) HRH3MCHR1LTA4HBACE1CYP2D6
SCHEMBL14039753 0.81 MCHR1 (0.78) HRH3MCHR1LTA4HCYP2D6CHRM1
SCHEMBL12440251 0.81 MCHR1 (0.78) HRH3MCHR1LTA4HCYP2D6CHRM1
SCHEMBL12440472 0.80 MCHR1 (0.77) HRH3MCHR1LTA4HCYP2D6CHRM1
SCHEMBL2322941 0.80 MCHR1 (0.71) MCHR1CYP2D6CHRM1HTR2A
SCHEMBL12441623 0.79 MAP4K4 (0.60) HRH3MCHR1LTA4HBACE1CYP2D6
SCHEMBL12440309 0.79 MCHR1 (0.76) HRH3MCHR1LTA4HCYP2D6CHRM1
SCHEMBL12440372 0.79 MCHR1 (0.74) HRH3MCHR1LTA4HCYP2D6CHRM1
SCHEMBL21462645 0.78 HRH3 (0.86) HRH3LTA4HBACE1HRH1KCNH2
SCHEMBL12440442 0.78 MCHR1 (0.65) MCHR1LTA4HCYP2D6CHRM1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed