SCHEMBL12440639

SCHEMBL12440639

Clc1ccc(-c2ccc(-c3ccc4c(ccn4CCN4CCCC4)c3)nc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 12/20 0.48
HTR7 P34969 3/20 0.46
HTR6 P50406 2/20 0.42
CYP2D6 P10635 1/20 0.41
CHRM1 P11229 1/20 0.41
HTR2A P28223 1/20 0.41
CNR2 P34972 1/20 0.39
MET P08581 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440204 0.89 MCHR1 (0.39) MCHR1HTR7HTR6CHRM1HTR2A
SCHEMBL14767425 0.89 HTR7 (0.43) MCHR1HTR7HTR6MET
SCHEMBL12440514 0.87 HTR7 (0.39) MCHR1HTR7HTR6MET
SCHEMBL12441448 0.85 HRH3 (0.44) MCHR1HTR7HTR2AMET
SCHEMBL13933553 0.82 MCHR1 (0.65) MCHR1
SCHEMBL12440000 0.82 MCHR1 (0.46) MCHR1CYP2D6CHRM1HTR2ACNR2
SCHEMBL2319646 0.81 MCHR1 (0.62) MCHR1CYP2D6CHRM1HTR2A
SCHEMBL23927826 0.79 HTR7 (0.63) HTR7HTR6HTR2A
SCHEMBL12440655 0.78 NPY5R (0.37)
SCHEMBL12441321 0.78 SCN9A (0.39) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2357173-A1 New alkyne compounds with MCH-antagonistic activity and medicaments containing them Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-08-17 EP disclosed