SCHEMBL14767425

SCHEMBL14767425

Nc1ccc(-c2ccc(-c3ccc4c(ccn4CCN4CCCC4)c3)nc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 7/20 0.43
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
MCHR1 Q99705 2/20 0.39
MET P08581 1/20 0.39
HTR6 P50406 2/20 0.38
ESRRG P62508 2/20 0.37
HRH3 Q9Y5N1 3/20 0.37
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12440639 0.89 MCHR1 (0.48) HTR7MCHR1METHTR6
SCHEMBL215782 0.79 HTR7 (0.56) HTR7NOS3NOS1NOS2ESRRG
SCHEMBL12440204 0.79 MCHR1 (0.39) HTR7MCHR1METHTR6HRH3
SCHEMBL4263907 0.78 HTR7 (0.54) HTR7NOS3NOS1NOS2HTR6
SCHEMBL2262498 0.78 HTR7 (0.54) HTR7NOS3NOS1NOS2HTR6
SCHEMBL12440514 0.77 HTR7 (0.39) HTR7MCHR1METHTR6
SCHEMBL20784089 0.76 HTR7 (0.59) HTR7NOS3NOS1NOS2
SCHEMBL20604809 0.75 HTR7 (0.49) HTR7NOS3NOS1NOS2MET
SCHEMBL12441448 0.74 HRH3 (0.44) HTR7MCHR1METHRH3
SCHEMBL14767429 0.73 MCHR1 (0.46) NOS3NOS1NOS2MCHR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-B1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA (DE) 2013-03-13 EP disclosed