SCHEMBL12445781

SCHEMBL12445781

C=C(C)COc1cnc(C(=O)Nc2ccc(F)c(CCC(=O)NC)c2)cn1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.47
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
BACE2 Q9Y5Z0 8/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446234 0.84 BACE1 (0.47) BACE1NPC1RAB9ASMN1; SMN2BACE2
SCHEMBL12446154 0.83 BACE1 (0.54) BACE1
SCHEMBL7940427 0.79 SMN1; SMN2 (0.48) BACE1NPC1RAB9ASMN1; SMN2BACE2
SCHEMBL7942651 0.78 BACE1 (0.47) BACE1NPC1RAB9ASMN1; SMN2BACE2
SCHEMBL7943975 0.77 BACE1 (0.61) BACE1BACE2CYP2D6CYP2C9KCNH2
SCHEMBL12446185 0.75 NPC1 (0.43) BACE1NPC1RAB9ASMN1; SMN2BACE2
SCHEMBL12445581 0.74 BACE1 (0.56) BACE1BACE2
SCHEMBL17277723 0.73 BACE1 (0.56) BACE1BACE2KCNH2
SCHEMBL7942653 0.73 BACE1 (0.46) BACE1NPC1RAB9ASMN1; SMN2BACE2
SCHEMBL7942303 0.73 NPC1 (0.53) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed