SCHEMBL7942653

SCHEMBL7942653

CNC(=O)CCc1cc(NC(=O)c2ncc(F)cc2F)ccc1F

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.46
BACE2 Q9Y5Z0 6/20 0.45
GRM4 Q14833 3/20 0.43
KCNH2 Q12809 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17277722 0.85 BACE1 (0.52) BACE1BACE2GRM4KCNH2NPC1
SCHEMBL7933959 0.83 BACE1 (0.48) BACE1BACE2
SCHEMBL7940427 0.80 SMN1; SMN2 (0.48) BACE1BACE2GRM4NPC1RAB9A
SCHEMBL7942651 0.79 BACE1 (0.47) BACE1BACE2NPC1RAB9ASMN1; SMN2
SCHEMBL15443906 0.77 BACE1 (0.53) BACE1BACE2GRM4NPC1RAB9A
SCHEMBL7942303 0.76 NPC1 (0.53) NPC1RAB9ASMN1; SMN2
SCHEMBL14734050 0.75 BACE1 (0.50) BACE1BACE2NPC1RAB9ASMN1; SMN2
SCHEMBL7941769 0.74 POLB (0.54) BACE1NPC1RAB9ASMN1; SMN2
SCHEMBL8027585 0.73 MPO (0.50) RAB9ASMN1; SMN2
SCHEMBL7942306 0.73 MEN1 (0.51) GRM4NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010047372-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY 塩野義製薬株式会社 (JP) 2010-04-29 WO disclosed