SCHEMBL12445978

SCHEMBL12445978

Nc1ncccc1NCc1cc(NC(=O)c2cnc(OCC#CCF)cn2)ccn1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.65
BACE2 Q9Y5Z0 4/20 0.41
CTSD P07339 1/20 0.39
CYP2D6 P10635 1/20 0.38
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7946763 0.92 BACE1 (0.66) BACE1BACE2CTSDAPP
SCHEMBL12445787 0.92 BACE1 (0.66) BACE1BACE2CTSDAPP
SCHEMBL7944986 0.92 BACE1 (0.68) BACE1BACE2CTSDAPP
SCHEMBL12445909 0.92 BACE1 (0.68) BACE1BACE2APP
SCHEMBL7940563 0.91 BACE1 (0.65) BACE1BACE2CTSDAPP
SCHEMBL12445765 0.91 BACE1 (0.79) BACE1BACE2CTSDAPP
SCHEMBL7945386 0.89 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL12446306 0.88 BACE1 (0.83) BACE1BACE2CTSD
SCHEMBL7941611 0.88 BACE1 (0.65) BACE1BACE2CYP2D6
SCHEMBL7942740 0.87 BACE1 (0.64) BACE1BACE2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed