SCHEMBL1245684

SCHEMBL1245684

C[n+]1ccc(C=Cc2ccc(NC(=O)[C@@H](N)CCC(=O)O)cc2)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHAT P28329 2/20 0.53
APP P05067 3/20 0.48
RAD52 P43351 3/20 0.47
LTA4H P09960 5/20 0.46
PKM P14618 3/20 0.44
HTT P42858 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 2/20 0.44
NPC1 O15118 2/20 0.44
NSD2 O96028 2/20 0.44
POLB P06746 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MAPT P10636 2/20 0.42
MAPK1 P28482 2/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
BACE1 P56817 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1246932 0.89 CHAT (0.53) CHATAPPRAD52LTA4HPKM
SCHEMBL1245825 0.88 CHAT (0.49) CHATAPPRAD52PKMHTT
SCHEMBL1245828 0.86 CHAT (0.53) CHATAPPRAD52LTA4HPKM
SCHEMBL1245827 0.86 LTA4H (0.48) CHATRAD52LTA4HPKMHTT
Hydrochloric Acid SCHEMBL1244769 0.85 CHAT (0.51) CHATAPPRAD52PKMHTT
SCHEMBL1245863 0.85 CHAT (0.57) CHATAPPRAD52LTA4HPKM
Hydrochloric Acid SCHEMBL1246494 0.82 BACE1 (0.56) CHATAPPRAD52PKMHTT
Hydrochloric Acid SCHEMBL1244753 0.81 CHAT (0.53) CHATAPPRAD52LTA4HPKM
SCHEMBL1246509 0.80 CHAT (0.52) CHATAPPRAD52LTA4HPKM
SCHEMBL1246159 0.80 CHAT (0.51) CHATAPPRAD52LTA4HPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459734-A2 NOVEL PEPTIDASE SUBSTRATES Biomérieux (FR) 2012-06-06 EP claimed
WO-2011012809-A2 NOVEL PEPTIDASE SUBSTRATES bioMérieux (FR) 2011-02-03 WO claimed
EP-2459734-A2 NOVEL PEPTIDASE SUBSTRATES Biomérieux (FR) 2012-06-06 EP disclosed
WO-2011012809-A2 NOVEL PEPTIDASE SUBSTRATES bioMérieux (FR) 2011-02-03 WO disclosed