SCHEMBL124592

SCHEMBL124592

O=C(O)c1cnc2ncccc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.59
PSMD14 O00487 2/20 0.55
KDM4E B2RXH2 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
LMNA P02545 1/20 0.50
ACP1 P24666 1/20 0.46
HCAR2 Q8TDS4 2/20 0.44
ALDH1A1 P00352 2/20 0.44
APP P05067 1/20 0.44
GAA P10253 1/20 0.44
HCAR3 P49019 1/20 0.44
PDE4A P27815 1/20 0.43
P4HA1 P13674 3/20 0.41
P4HTM Q9NXG6 2/20 0.41
KDM6B O15054 1/20 0.41
KDM4A O75164 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM2A Q9Y2K7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30392839 1.00 MGAM (0.59) MGAMPSMD14KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL7010614 0.98 MGAM (0.57) MGAMPSMD14KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL9378228 0.98 MGAM (0.57) MGAMPSMD14KDM4EMEN1KMT2A
Water SCHEMBL8227338 0.89 ACP1 (0.51) MGAMPSMD14KDM4EMEN1KMT2A
SCHEMBL28015646 0.86 PSMD14 (0.47) MGAMPSMD14KDM4EMEN1KMT2A
SCHEMBL27501111 0.85 MGAM (0.79) MGAMPSMD14KDM4EMEN1KMT2A
SCHEMBL163182 0.84 PSMD14 (0.56) MGAMPSMD14KDM4EMEN1KMT2A
Aspartic Acid SCHEMBL27878589 0.84 MGAM (0.43) MGAMPSMD14KDM4EMEN1KMT2A
Hydrochloric Acid SCHEMBL14966721 0.83 PSMD14 (0.55) MGAMPSMD14KDM4EMEN1KMT2A
SCHEMBL21358078 0.83 PSMD14 (0.60) MGAMPSMD14KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 520 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113825756-A Substituted polycyclic carboxylic acids, analogs thereof, and methods of use thereof 爱彼特生物制药公司 2021-12-21 CN claimed
CN-110475777-A For treating and preventing new pyrido [2,3-b] benzazolyl compounds of bacterium infection HOFFMANN LA ROCHE 2019-11-19 CN claimed
CN-107286182-A Novel oxazolidinone fluoro quinolone derivative and purposes 李靖 2017-10-24 CN claimed
CN-106632317-A 1,4-dihydro-naphthyridine derivative and pharmaceutical composition and application thereof 江苏欧威医药有限公司 2017-05-10 CN claimed
CN-104203945-B 1, 4-dihydro-naphthyridine derivatives, pharmaceutical compositions and uses thereof 江苏欧威医药有限公司 2017-01-18 CN claimed
CN-105481851-A Hexahydrobenzonaphthyridine-type optically active compound and pharmaceutical use thereof ZHAOLONG GONG 2016-04-13 CN claimed
WO-2007028171-A9 METHODS OF USING (+)-1,4-DIHYDRO-7-[(3S,4S)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID FOR TREATMENT OF CANCER SUNESIS PHARMACEUTICALS, INC. (US) 2014-12-11 WO claimed
CN-104203945-A 1, 4-dihydro-naphthyridine derivatives, pharmaceutical compositions and uses thereof JIANGSU SIMOVAY PHARMACEUTICAL CO LTD 2014-12-10 CN claimed
CN-103889414-A pharmaceutical composition RAQUALIA PHARMA INC 2014-06-25 CN claimed
CN-102574840-B R-7-(3-aminomethyl-4-methoxyimino-3-methyl-pyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid and l-aspartic acid salt, process for the preparation thereof and pharmaceutical composition comprising the same ARMED INC 2014-05-28 CN claimed
CN-1377347-A Pharmaceutically active sulfonamide derivatives APPLIED RESEARCH SYSTEMS (NL) 2002-10-30 CN claimed
EP-1230235-A1 COMPOUNDS WITH ANTIBACTERIAL AND ANTIPARASITIC PROPERTIES New Pharma Research Sweden AB (SE) 2002-08-14 EP claimed
WO-2001036408-A1 COMPOUNDS WITH ANTIBACTERIAL AND ANTIPARASITIC PROPERTIES NEW PHARMA RESEARCH SWEDEN AB (SE) 2001-05-25 WO claimed
CN-1257489-A Substituted benzopyran derivatives for the treatment of inflammation SEARLE & CO (US) 2000-06-21 CN claimed
WO-1995007909-A1 ALKYL-1-ALKYL-4-HYDROXY-2-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLATES AS ANTI-RHEUMATIC AGENTS KNOLL AG (DE) 1995-03-23 WO claimed
EP-0562042-A4 QUINOLINE, NAPHTHYRIDINE AND PYRIDOBENZOXAZINE DERIVATIVES ABBOTT LAB (US) 1994-07-06 EP claimed
EP-0562042-A1 QUINOLINE, NAPHTHYRIDINE AND PYRIDOBENZOXAZINE DERIVATIVES ABBOTT LABORATORIES (US) 1993-09-29 EP claimed
WO-1992010191-A1 QUINOLINE, NAPHTHYRIDINE AND PYRIDOBENZOXAZINE DERIVATIVES ABBOTT LABORATORIES (US) 1992-06-25 WO claimed
EP-0120832-B1 4-ALKYLINDOLONAPHTHYRIDINES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM OMNICHEM Société anonyme (BE) 1987-04-29 EP claimed
EP-0120832-A1 4-Alkylindolonaphthyridines and pharmaceutical compositions containing them OMNICHEM Société anonyme (BE) 1984-10-03 EP claimed