SCHEMBL12460552

SCHEMBL12460552

CCO[C@H]1C[C@H](COS(=O)(=O)c2ccc(C)cc2)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.40
MMP13 P45452 1/20 0.40
MCL1 Q07820 4/20 0.39
GPR119 Q8TDV5 7/20 0.39
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ABCB1 P08183 1/20 0.37
GAA P10253 1/20 0.36
TSHR P16473 1/20 0.36
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29105266 0.89 CYP2D6 (0.42) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL29765023 0.89 CYP2D6 (0.42) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL8015585 0.89 CYP2D6 (0.42) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL1366652 0.89 CYP2D6 (0.42) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL1366650 0.89 CYP2D6 (0.42) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL22207663 0.87 ABCB1 (0.51) MCL1GPR119ABCB1
SCHEMBL21996502 0.87 ABCB1 (0.51) MCL1GPR119ABCB1
SCHEMBL9067588 0.87 ABCB1 (0.51) MCL1GPR119ABCB1
SCHEMBL12460550 0.86 CYP2D6 (0.39) HSD11B1MMP13MCL1GPR119CYP1A2
SCHEMBL21996496 0.86 GPR119 (0.43) MCL1GPR119MEN1KMT2AABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343286-A1 Dibenzo[b,f][1,4]oxazepine derivatives as inhibitors of histone deacetylase Methylgene, Inc. (CA) 2011-07-13 EP disclosed