SCHEMBL1246424

SCHEMBL1246424

Cc1onc(-c2ccc(-c3cc(C(=O)O)ccn3)cc2)c1NC(=O)OCCc1ccccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.52
SCN5A Q14524 6/20 0.52
KDM4C Q9H3R0 4/20 0.44
KDM5A P29375 1/20 0.44
KDM5B Q9UGL1 1/20 0.44
KMO O15229 1/20 0.40
NTRK1 P04629 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 2/20 0.37
MAPT P10636 1/20 0.37
KDM4A O75164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1245322 0.89 SCN9A (0.57) SCN9ASCN5ANTRK1TDP1GAA
SCHEMBL1247566 0.88 SCN9A (0.59) SCN9ASCN5ANTRK1GAAMAPT
SCHEMBL1247099 0.87 SCN9A (0.53) SCN9ASCN5ANTRK1
SCHEMBL3714247 0.87 LPAR1 (0.46) SCN9ASCN5AKDM4CKDM5AKDM5B
SCHEMBL1247125 0.86 SCN9A (0.58) SCN9ASCN5ANTRK1TDP1GAA
SCHEMBL1246240 0.86 SCN9A (0.54) SCN9ASCN5ANTRK1TDP1GAA
SCHEMBL1245113 0.85 SCN9A (0.54) SCN9ASCN5ATDP1MAPT
SCHEMBL1247223 0.85 SCN9A (0.52) SCN9ASCN5ANTRK1TDP1GAA
SCHEMBL1246291 0.84 SCN9A (0.57) SCN9ASCN5ANTRK1TDP1GAA
SCHEMBL1247808 0.84 SCN9A (0.56) SCN9ASCN5ANTRK1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed