SCHEMBL12466322

SCHEMBL12466322

Fc1cccc(CNc2ccnc(-c3ccnc(F)c3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.46
CLK1 P49759 2/20 0.46
KDM5A P29375 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
KDM5B Q9UGL1 1/20 0.45
HPGD P15428 2/20 0.43
NTRK1 P04629 1/20 0.42
NTRK3 Q16288 1/20 0.42
NTRK2 Q16620 1/20 0.42
MAP4K4 O95819 2/20 0.42
GSK3B P49841 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
AURKA O14965 1/20 0.42
DAPK3 O43293 1/20 0.42
JAK2 O60674 1/20 0.42
PRKD3 O94806 1/20 0.42
PAK4 O96013 1/20 0.42
ABL1 P00519 1/20 0.42
LCK P06239 1/20 0.42
CSF1R P07333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12466193 0.82 KDM5A (0.52) DYRK1ACLK1KDM5AKDM4CKDM5B
SCHEMBL1461900 0.81 CCNT1 (0.55) KDM5AKDM4CKDM5BCCNT1
SCHEMBL6122655 0.80 CCNT1 (0.53) DYRK1ACLK1KDM5AKDM4CKDM5B
SCHEMBL1191606 0.78 CCNT1 (0.64) KDM5AKDM4CKDM5BKDRCCNT1
SCHEMBL12466070 0.78 CCNT1 (0.69) CCNT1CDK9
SCHEMBL12466282 0.77 KDM5A (0.50) DYRK1ACLK1KDM5AKDM4CKDM5B
SCHEMBL1191651 0.76 CCNT1 (0.68) KDM5AKDM4CKDM5BMAP4K4GSK3B
SCHEMBL27876840 0.74 F2 (0.51) KCNH3KDM4EGAA
SCHEMBL6696141 0.74 HPGD (0.60) KDM5AKDM4CKDM5BHPGDFFAR1
SCHEMBL6229701 0.74 HPGD (0.65) HPGDFFAR1CDK2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101066-A1 PYRIDINE BIARYL AMINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed
WO-2012101065-A2 PYRIMIDINE BIARYL AMINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed