SCHEMBL12466282

SCHEMBL12466282

Fc1cccc(CNc2ccnc(Cl)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.50
KDM4C Q9H3R0 1/20 0.50
KDM5B Q9UGL1 1/20 0.50
HPGD P15428 1/20 0.48
CCNT1 O60563 7/20 0.48
CDK9 P50750 5/20 0.48
FFAR1 O14842 1/20 0.46
NTRK1 P04629 3/20 0.46
NTRK3 Q16288 1/20 0.46
NTRK2 Q16620 1/20 0.46
P2RX7 Q99572 1/20 0.45
NOS1 P29475 1/20 0.45
DYRK1A Q13627 2/20 0.45
CLK1 P49759 1/20 0.45
MAOB P27338 1/20 0.44
HTR6 P50406 1/20 0.44
CLK4 Q9HAZ1 2/20 0.44
AURKA O14965 1/20 0.43
DAPK3 O43293 1/20 0.43
JAK2 O60674 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4646979 0.83 KDM4E (0.47) HPGDCCNT1CDK9NTRK1NTRK3
SCHEMBL27893661 0.83 GRIN2D (0.49)
SCHEMBL6756755 0.82 GHSR (0.46) MAOBHTR6AURKAABL1
SCHEMBL6229701 0.79 HPGD (0.65) HPGDFFAR1NOS1MAOB
SCHEMBL6696141 0.79 HPGD (0.60) KDM5AKDM4CKDM5BHPGDFFAR1
SCHEMBL6692696 0.77 FFAR1 (0.67) KDM5AKDM4CKDM5BHPGDFFAR1
SCHEMBL12466322 0.77 DYRK1A (0.46) KDM5AKDM4CKDM5BHPGDCCNT1
SCHEMBL6754268 0.77 MAPT (0.56)
SCHEMBL12466337 0.77 CCNT1 (0.57) KDM5AKDM4CKDM5BCCNT1DYRK1A
SCHEMBL15378645 0.75 CLK4 (0.46) KDM5AKDM4CKDM5BCCNT1NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101065-A2 PYRIMIDINE BIARYL AMINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed
WO-2012101066-A1 PYRIDINE BIARYL AMINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed