SCHEMBL12469102

SCHEMBL12469102

O=C(Nc1ccncc1)c1cccc(N2CC[C@@H](NCC3CCN(C4CCCC4)C3)C2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 7/20 0.41
PRKCQ Q04759 2/20 0.37
S1PR1 P21453 2/20 0.37
OGFRL1 Q5TC84 1/20 0.37
KDR P35968 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
STAT3 P40763 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
IRAK4 Q9NWZ3 2/20 0.35
TTR P02766 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12685439 1.00 HSD11B1 (0.41) HSD11B1PRKCQS1PR1OGFRL1KDR
SCHEMBL12685434 1.00 HSD11B1 (0.41) HSD11B1PRKCQS1PR1OGFRL1KDR
SCHEMBL12469347 0.96 HSD11B1 (0.42) HSD11B1PRKCQS1PR1OGFRL1KDR
SCHEMBL12469060 0.84 FLT3 (0.42) HSD11B1PRKCQIRAK4CA12CA1
SCHEMBL12468994 0.83 NAMPT (0.39) HSD11B1PRKCQIRAK4CA12CA1
SCHEMBL12469124 0.83 NAMPT (0.39) HSD11B1PRKCQIRAK4CA12CA1
SCHEMBL19222529 0.79 HSD11B1 (0.37) HSD11B1PRKCQOGFRL1HRH3IRAK4
SCHEMBL19222456 0.79 HSD11B1 (0.37) HSD11B1PRKCQOGFRL1HRH3IRAK4
SCHEMBL15347563 0.77 HSD11B1 (0.50) HSD11B1KDRHRH3ALDH1A1LMNA
SCHEMBL30077118 0.77 HSD11B1 (0.50) HSD11B1KDRHRH3ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627649-A1 CXCR4 RECEPTOR ANTAGONISTS Proximagen Limited (GB) 2013-08-21 EP disclosed
WO-2012049277-A1 CXCR4 RECEPTOR ANTAGONISTS PROXIMAGEN LTD (GB) 2012-04-19 WO disclosed