SCHEMBL12469284

SCHEMBL12469284

C=C(C(=O)O)C(O)c1ccc(Cl)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
APP P05067 2/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
S1PR3 Q99500 6/20 0.40
S1PR1 P21453 4/20 0.40
FFAR1 O14842 1/20 0.39
HPGD P15428 1/20 0.38
KCNQ3 O43525 2/20 0.37
KCNQ2 O43526 2/20 0.37
KCNE1 P15382 2/20 0.37
KCNQ1 P51787 2/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
KMO O15229 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12468991 0.87 MDM2 (0.43) CES2CES1S1PR3S1PR1HPGD
SCHEMBL12469122 0.85 KEAP1 (0.42) HPGDKMOSLC6A2SLC6A4SLC6A3
SCHEMBL23973484 0.83 APP (0.48) CES2CES1APPPSEN1PSEN2
SCHEMBL1280792 0.82 S1PR3 (0.39) CES2CES1APPPSEN1PSEN2
SCHEMBL12497587 0.78 CES2 (0.45) CES2CES1APPPSEN1PSEN2
SCHEMBL12499078 0.78 CES2 (0.45) CES2CES1APPPSEN1PSEN2
SCHEMBL28795492 0.75 HPGD (0.48) HPGD
SCHEMBL28795451 0.75 HPGD (0.48) CES2CES1HPGD
SCHEMBL18987936 0.75 MAPT (0.48) S1PR3HPGDPPARGPPARA
SCHEMBL16877159 0.73 PSEN1 (0.37) CES2CES1APPPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2625170-A1 1,4-OXAZEPANE DERIVATIVES Takeda Pharmaceutical Company Limited (JP) 2013-08-14 EP disclosed
WO-2012046882-A1 1,4-OXAZEPANE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-04-12 WO disclosed