SCHEMBL12469575

SCHEMBL12469575

CCCc1c[nH]c(-c2ccccn2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
PKM P14618 2/20 0.41
ALPL P05186 2/20 0.41
ALOX15 P16050 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
HSD17B10 Q99714 1/20 0.41
CBFB Q13951 4/20 0.41
METAP1 P53582 6/20 0.41
METAP2 P50579 5/20 0.41
LMNA P02545 3/20 0.41
HPGD P15428 1/20 0.41
MTOR P42345 1/20 0.41
PDPK1 O15530 1/20 0.40
KDM4E B2RXH2 4/20 0.40
CCR1 P32246 2/20 0.39
CCR5 P51681 2/20 0.39
CCR8 P51685 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619864 0.90 PDPK1 (0.44) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL19691749 0.81 CBFB (0.49) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL18091913 0.79 F2 (0.43) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL11303973 0.77 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL535052 0.77 PDE5A (0.44) SMN1; SMN2NPC1RAB9APKMHSD17B10
SCHEMBL3327100 0.75 KDM4E (0.49) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL8311607 0.74 KDM4E (0.56) SMN1; SMN2NPC1RAB9ATDP1PKM
Dipyridyl SCHEMBL9115752 0.74 KDM4E (0.56) SMN1; SMN2NPC1RAB9ATDP1PKM
SCHEMBL29008471 0.74 TSHR (0.37) NPC1RAB9ATDP1ALOX15LMNA
Carbamic Acid SCHEMBL7648295 0.73 PDE4B (0.39) SMN1; SMN2NPC1RAB9ATDP1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627649-A1 CXCR4 RECEPTOR ANTAGONISTS Proximagen Limited (GB) 2013-08-21 EP disclosed
WO-2012049277-A1 CXCR4 RECEPTOR ANTAGONISTS PROXIMAGEN LTD (GB) 2012-04-19 WO disclosed