SCHEMBL12469680

SCHEMBL12469680

COc1cc(NCc2ccc(CN)cc2)c2ncccc2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.69
HDAC6 Q9UBN7 1/20 0.69
HSP90AA1 P07900 7/20 0.65
HSP90AB1 P08238 7/20 0.65
MEN1 O00255 5/20 0.63
KMT2A Q03164 5/20 0.63
KDM4E B2RXH2 3/20 0.63
MAPT P10636 2/20 0.63
L3MBTL1 Q9Y468 1/20 0.63
ALDH1A1 P00352 4/20 0.58
HTT P42858 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
TDP1 Q9NUW8 2/20 0.57
TDP2 O95551 1/20 0.57
FGB P02675 1/20 0.57
POLB P06746 1/20 0.57
GAA P10253 1/20 0.57
THRB P10828 1/20 0.57
TSHR P16473 1/20 0.57
NR4A1 P22736 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30996045 0.81 MAPT (0.62) HDAC1HDAC6MEN1KMT2AKDM4E
SCHEMBL31020169 0.80 KMT2A (0.69) HDAC1HDAC6HSP90AA1HSP90AB1MEN1
SCHEMBL17792862 0.80 HSP90AA1 (0.93) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL21855430 0.80 KMT2A (0.69) HDAC1HDAC6HSP90AA1HSP90AB1MEN1
SCHEMBL8893299 0.79 HSP90AA1 (1.00) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL12470224 0.79 PKM (0.59) HDAC1HDAC6HSP90AA1HSP90AB1MEN1
SCHEMBL8891233 0.78 HSP90AA1 (0.98) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL8900580 0.78 HSP90AA1 (0.98) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL8891243 0.78 HSP90AA1 (0.98) HSP90AA1HSP90AB1MEN1KMT2AKDM4E
SCHEMBL8891533 0.78 HSP90AA1 (0.98) HSP90AA1HSP90AB1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012048894-A1 HYBRID COMPOUNDS OF 4- AND 8-AMINOQUINOLINES FOR THE PROPHYLACTIC AND THERAPEUTIC TREATMENT OF MALARIA AND OTHER PARASITIC DISEASES JULIUS-MAXIMILIANS-UNIVERSITÄT WÜRZBURG (DE) 2012-04-19 WO disclosed