SCHEMBL31020169

SCHEMBL31020169

COc1cc(NCc2ccccn2)c2ncccc2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.69
MEN1 O00255 5/20 0.69
KDM4E B2RXH2 3/20 0.69
MAPT P10636 2/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
HSP90AA1 P07900 7/20 0.61
HSP90AB1 P08238 7/20 0.61
ALDH1A1 P00352 3/20 0.60
HDAC1 Q13547 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
TDP1 Q9NUW8 3/20 0.57
POLB P06746 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
TDP2 O95551 1/20 0.57
FGB P02675 1/20 0.57
GAA P10253 1/20 0.57
THRB P10828 1/20 0.57
TSHR P16473 1/20 0.57
NR4A1 P22736 1/20 0.57
HTT P42858 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21855430 1.00 KMT2A (0.69) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL12469680 0.80 HDAC1 (0.69) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL31020173 0.78 MEN1 (0.62) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL11812974 0.78 KMT2A (0.61) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL17714697 0.77 KMT2A (0.53) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL9850421 0.77 HSP90AA1 (0.65) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL18163920 0.77 HSP90AA1 (0.80) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL13856507 0.77 HSP90AA1 (0.80) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL17792862 0.77 HSP90AA1 (0.93) KMT2AMEN1KDM4EMAPTL3MBTL1
SCHEMBL18292338 0.76 MAOA (0.60) KMT2AMEN1KDM4EMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3866802-B1 QUINONE REDUCTASE 2 INHIBITORS FOR USE AS NEUROPROTECTIVE AGENTS UNIV DUKE (US) 2024-08-21 EP claimed
CN-112823006-B Quinone reductase 2 inhibitors as neuroprotective agents 杜克大学 2024-09-17 CN disclosed