SCHEMBL1246985

SCHEMBL1246985

CC(=O)Oc1ccc2c(c1)CCC1C2CC[C@]2(C)C=CCC12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.67
SMN1; SMN2 Q16637 4/20 0.67
ESR1 P03372 4/20 0.67
ADORA3 P0DMS8 2/20 0.67
ATM Q13315 2/20 0.67
PGR P06401 2/20 0.67
SLC6A3 Q01959 2/20 0.67
AR P10275 1/20 0.67
CHRM1 P11229 1/20 0.67
TBXA2R P21731 1/20 0.67
ADRA1A P35348 1/20 0.67
OPRM1 P35372 1/20 0.67
CYP3A4 P08684 4/20 0.64
MAPT P10636 3/20 0.64
TP53 P04637 1/20 0.64
STS P08842 2/20 0.52
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
NR3C1 P04150 2/20 0.52
SLC6A2 P23975 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4284331 1.00 LMNA (0.67) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL1248414 0.89 MAPT (0.66) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL4281651 0.89 MAPT (0.66) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL7596856 0.87 SMN1; SMN2 (0.53) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL5679838 0.86 LMNA (0.64) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL5154685 0.86 LMNA (0.64) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL1246984 0.86 LMNA (0.64) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL5679791 0.86 LMNA (0.64) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL5682148 0.86 LMNA (0.64) LMNASMN1; SMN2ESR1ADORA3ATM
SCHEMBL8518252 0.85 ESR1 (0.48) LMNASMN1; SMN2ESR1ADORA3ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278880-A1 STEROID TREATMENT FOR HOT FLASHES Pherin Pharmaceuticals, Inc. (US) 2011-02-02 EP claimed
US-20090258040-A1 STEROID TREATMENT FOR HOT FLASHES PHERIN PHARMACEUTICALS, INC. (US) 2009-10-15 US claimed
WO-2009126825-A1 STEROID TREATMENT FOR HOT FLASHES PHERIN PHARMACEUTICALS, INC. (US) 2009-10-15 WO claimed
EP-1251856-B1 METHOD OF INCREASING ALERTNESS BY ADMINISTRATION OF A VOMEROPHERIN, AND VOMEROPHERIN-EMITTING ALARM DEVICES PHERIN PHARM INC (US) 2005-06-15 EP claimed
EP-0891188-A4 STEROIDS AS NEUROCHEMICAL INITIATORS OF CHANGE IN HUMAN BLOOD LEVELS OF LH OR FSH PHERIN PHARM INC (US) 2004-09-01 EP claimed
US-6544971-B1 Alarm device especially for detecting fires, unauthorized entry or sleep apnea, or the presence of CO, CH4, propane or radon PHERIN PHARMACEUTICALS, INC. 2003-04-08 US claimed
EP-1251856-A1 METHOD OF INCREASING ALERTNESS BY ADMINISTRATION OF A VOMEROPHERIN, AND VOMEROPHERIN-EMITTING ALARM DEVICES Pherin Pharmaceuticals, Inc. (US) 2002-10-30 EP claimed
US-6331534-B1 ADMINISTERING EFFECTIVE AMOUNT OF STEROID WITHIN NASAL PASSAGE OF INDIVIDUAL SUCH THAT IT BINDS SPECIFICALLY TO RECEPTORS ON SURFACE OF NASAL NEUROEPITHELIAL CELLS IN VOMERONASAL ORGAN PHERIN PHARMACEUTICALS, INC. 2001-12-18 US claimed
WO-2001056577-A1 METHOD OF INCREASING ALERTNESS BY ADMINISTRATION OF A VOMEROPHERIN, AND VOMEROPHERIN-EMITTING ALARM DEVICES PHERIN PHARMACEUTICALS, INC. (US) 2001-08-09 WO claimed
EP-0715517-A4 ESTRENE STEROIDS AS NEUROCHEMICAL INITIATORS OF CHANGE IN HUMAN HYPOTHALAMIC FUNCTION AND RELATED PHARMACEUTICAL COMPOSITIONS AND METHODS PHERIN CORP (US) 2000-10-11 EP claimed
JP-2000504025-A 2000-04-04 JP claimed
EP-0891188-A1 STEROIDS AS NEUROCHEMICAL INITIATORS OF CHANGE IN HUMAN BLOOD LEVELS OF LH OR FSH Pherin Pharmaceuticals, Inc. (US) 1999-01-20 EP claimed
US-5783571-A SUBSTITUTED TETRAENE STEROIDS FOR CONTROLLING GLANDULAR FUNCTION PHERIN CORPORATION (US) 1998-07-21 US claimed
EP-0715517-A1 ESTRENE STEROIDS AS NEUROCHEMICAL INITIATORS OF CHANGE IN HUMAN HYPOTHALAMIC FUNCTION AND RELATED PHARMACEUTICAL COMPOSITIONS AND METHODS PHERIN CORPORATION (US) 1996-06-12 EP claimed
WO-1994028903-A1 ESTRENE STEROIDS AS NEUROCHEMICAL INITIATORS OF CHANGE IN HUMAN HYPOTHALAMIC FUNCTION AND RELATED PHARMACEUTICAL COMPOSITIONS AND METHODS PHERIN CORPORATION (US) 1994-12-22 WO claimed
WO-2025217067-A1 INTRANASAL DRUG DELIVERY SYSTEM VISTAGEN THERAPEUTICS, INC. (US) 2025-10-16 WO disclosed
US-20090258040-A1 STEROID TREATMENT FOR HOT FLASHES PHERIN PHARMACEUTICALS, INC. (US) 2009-10-15 US disclosed
US-5272134-A Fragrance compositions and other compositions which contain human pheromones EROX CORPORATION (US) 1993-12-21 US disclosed
WO-1993018742-A1 FRAGRANCE COMPOSITIONS AND OTHER COMPOSITIONS WHICH CONTAIN HUMAN PHEROMONES EROX CORPORATION (US) 1993-09-30 WO disclosed
EP-0562843-A2 Fragrance compositions and other compositions which contain human pheromones EROX CORPORATION (US) 1993-09-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090258040-A1 STEROID TREATMENT FOR HOT FLASHES CYP19A1, SHBG, HSD17B11 LMNA 2321/4885SMN1; SMN2 3611/4885ESR1 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.