SCHEMBL12470372

SCHEMBL12470372

O=C1C(c2cc3c(cc2O)OCO3)c2ccccc2N1Cc1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 6/20 0.54
SCN9A Q15858 3/20 0.50
ADK P55263 4/20 0.46
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HPGD P15428 1/20 0.41
CMA1 P23946 1/20 0.41
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL281432 0.84 SIRT1 (0.46) GSK3BSCN9AADKLMNAMAPT
SCHEMBL2994860 0.81 SCN9A (0.52) GSK3BSCN9AADKTSHRALDH1A1
SCHEMBL27707819 0.80 SCN9A (0.53) GSK3BSCN9ALMNAMAPTTSHR
SCHEMBL281812 0.80 SCN9A (0.53) SCN9ATSHRHPGD
SCHEMBL281216 0.80 SCN9A (0.53) GSK3BSCN9ALMNAMAPTTSHR
SCHEMBL19763099 0.80 SCN9A (0.48) GSK3BSCN9AADKTSHRALDH1A1
SCHEMBL18606884 0.79 SCN9A (0.51) GSK3BSCN9AADKHPGD
SCHEMBL281104 0.79 GSK3B (0.47) GSK3BSCN9AADKLMNAMAPT
SCHEMBL27728408 0.79 SCN9A (0.48) SCN9ATSHRALDH1A1KMT2ASMN1; SMN2
SCHEMBL281769 0.79 SCN9A (0.75) SCN9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012049555-A1 SPIROCYCLIC COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS LUPIN LIMITED (IN) 2012-04-19 WO disclosed