SCHEMBL12480913

SCHEMBL12480913

CC(C)(C)C1C(=O)c2ccccc2OC12CCNCC2

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.44
OPRD1 P41143 15/20 0.41
KCNH2 Q12809 11/20 0.41
OPRK1 P41145 6/20 0.41
CYP2D6 P10635 5/20 0.38
ALDH1A1 P00352 1/20 0.38
OPRM1 P35372 1/20 0.37
PLA2G1B P04054 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14919110 0.83 MAPT (0.42) ATM
SCHEMBL14972882 0.83 HTR2C (0.40)
SCHEMBL13339981 0.83 OPRD1 (0.43) ATMOPRD1KCNH2OPRK1CYP2D6
Hydrochloric Acid SCHEMBL3495476 0.82 OPRD1 (0.42) ATMOPRD1KCNH2OPRK1CYP2D6
SCHEMBL3837866 0.80 OPRD1 (0.42) ATMOPRD1KCNH2OPRK1CYP2D6
SCHEMBL2591939 0.78 OPRD1 (0.39) ATMOPRD1KCNH2OPRK1CYP2D6
SCHEMBL2589311 0.77 OPRD1 (0.44) OPRD1KCNH2OPRK1CYP2D6ALDH1A1
SCHEMBL12482165 0.75 MAOB (0.46) OPRD1KCNH2OPRK1CYP2D6ALDH1A1
SCHEMBL3457811 0.74 OPRD1 (0.45) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL7845728 0.72 OPRD1 (0.38) OPRD1KCNH2OPRK1CYP2D6OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675812-A1 CHROMAN - SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS Vertex Pharmaceuticals Incorporated (US) 2013-12-25 EP disclosed
WO-2012112743-A1 CHROMAN - SPIROCYCLIC PIPERIDINE AMIDES AS MODULATORS OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-08-23 WO disclosed