SCHEMBL12486551

SCHEMBL12486551

COc1cccc(CC2NCCc3ccsc32)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.53
DRD2 P14416 2/20 0.53
HTR7 P34969 2/20 0.53
EED O75530 1/20 0.44
OPRM1 P35372 2/20 0.41
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRB3 P13945 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
PTGS1 P23219 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486539 0.85 BCHE (0.45)
SCHEMBL12486031 0.83 SLC22A1 (0.43) DRD2ADRB2ADRB1TBXA2R
SCHEMBL12484520 0.82 BCHE (0.54)
SCHEMBL12485686 0.81 GID4 (0.46) DRD2OPRM1ADRB2
SCHEMBL4709300 0.81 SLC22A1 (0.59) ADRB2
SCHEMBL12485011 0.80 SLC22A1 (0.40) DRD2ADRB2
SCHEMBL12486091 0.79 KDM4E (0.60) OPRM1ADRB2ADRB1HTR1AADRA2A
SCHEMBL12485294 0.79 SLC22A1 (0.42) DRD2ADRB2
SCHEMBL8559156 0.79 PRCP (0.66) CHRM4DRD2HTR7OPRM1ADRB2
SCHEMBL4026022 0.77 BCHE (0.67)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012114252-A1 NOVEL INDOLE AND PYRROLOPYRIDINE AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-08-30 WO disclosed