SCHEMBL12486605

SCHEMBL12486605

O=C(NO)c1noc2c1CN(C(=O)C(=Cc1ccccc1)c1cccs1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 9/20 0.39
RAB9A P51151 9/20 0.39
HSP90AA1 P07900 2/20 0.38
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HDAC1 Q13547 1/20 0.36
MAPT P10636 5/20 0.35
CHRM1 P11229 1/20 0.35
GAA P10253 1/20 0.35
NFKB1 P19838 2/20 0.35
NFKB2 Q00653 2/20 0.35
RELA Q04206 2/20 0.35
CASP3 P42574 2/20 0.35
SENP7 Q9BQF6 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12486603 1.00 KMT2A (0.39) KMT2ASMN1; SMN2LMNAMEN1TSHR
SCHEMBL12684591 0.88 HPGD (0.47) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12486947 0.88 HPGD (0.47) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12486948 0.88 HPGD (0.47) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12486525 0.84 HPGD (0.41) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12684589 0.84 HPGD (0.41) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12486521 0.84 HPGD (0.41) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12485722 0.82 KMT2A (0.41) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12485727 0.82 KMT2A (0.41) KMT2ASMN1; SMN2LMNAMEN1NPC1
SCHEMBL12487063 0.78 RAB9A (0.42) KMT2ASMN1; SMN2LMNAMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012117421-A1 HISTONE DEACETYLASE INHIBITORS ORCHID RESEARCH LABORATORIES LTD (IN) 2012-09-07 WO claimed
WO-2012117421-A1 HISTONE DEACETYLASE INHIBITORS ORCHID RESEARCH LABORATORIES LTD (IN) 2012-09-07 WO disclosed