SCHEMBL1249929

SCHEMBL1249929

NC(=O)c1cc(Cl)c(O)c(Cl)c1-n1nnc2cc(C(=O)O)ccc21

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 17/20 0.45
HPGD P15428 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
KCNMA1 Q12791 1/20 0.42
RXRA P19793 1/20 0.41
PPARG P37231 1/20 0.41
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1250337 0.78 HCAR3 (0.48) HCAR3HPGDHCAR2KCNMA1RXRA
SCHEMBL5437652 0.69 HCAR3 (0.57) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL2490016 0.69 HCAR3 (0.60) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL1248894 0.68 HCAR3 (0.50) HCAR3HPGDHCAR2KCNMA1RXRA
SCHEMBL1250575 0.68 HCAR3 (0.50) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL7537331 0.67 HCAR3 (0.62) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL30864289 0.67 HCAR3 (0.57) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL24927222 0.66 HCAR3 (0.65) HCAR3HPGDHCAR2RXRAPPARG
SCHEMBL996446 0.65 GLA (0.45) HPGDKCNMA1
SCHEMBL5921944 0.65 HCAR3 (0.68) HCAR3HPGDHCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879893-B2 Zinc binding ligand; sustained release of insulin NOVO NORDISK A/S (DK) 2011-02-01 US disclosed