SCHEMBL12560010

SCHEMBL12560010

CCCCc1ccc2c(c1)C1(c3ccccc3-c3ccc(N(c4ccccc4)c4ccc5c(c4)c4ccccc4n5-c4ccccc4)cc31)c1cc(CCCC)ccc1-2

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDK2 Q15119 1/20 0.33
RORA P35398 1/20 0.33
RORC P51449 1/20 0.33
RORB Q92753 1/20 0.33
MCHR2 Q969V1 2/20 0.33
PLA2G4A P47712 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
GLA P06280 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
GPR3 P46089 1/20 0.30
FDFT1 P37268 1/20 0.30
CNR2 P34972 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12560036 0.95 PLA2G4A (0.35) PDK2RORARORCRORBMCHR2
SCHEMBL12560141 0.95 PDK2 (0.35) KDM4EATML3MBTL1PDK2RORA
SCHEMBL13634082 0.94 PDK2 (0.39) KDM4EATML3MBTL1PDK2MCHR2
SCHEMBL13634127 0.92 RORA (0.35) PDK2RORARORCRORBMCHR2
SCHEMBL12560002 0.91 PDK2 (0.37) KDM4EATML3MBTL1PDK2RORA
SCHEMBL13634083 0.89 PDK2 (0.38) KDM4EPDK2PLA2G4AALDH1A1CYP1A2
SCHEMBL13634120 0.89 PDK2 (0.41) KDM4EATML3MBTL1PDK2PLA2G4A
SCHEMBL18135001 0.88 KDM4E (0.43) KDM4EATML3MBTL1PDK2
SCHEMBL29373143 0.88 KDM4E (0.43) KDM4EATML3MBTL1PDK2
SCHEMBL25563166 0.88 KDM4E (0.43) KDM4EATML3MBTL1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2018-06-21 US disclosed
US-9899602-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2018-02-20 US disclosed
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2017-05-04 US disclosed
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2017-05-04 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-9203035-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (KE) 2015-12-01 US disclosed
US-9203035-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (KE) 2015-12-01 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
US-20110147728-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2011-06-23 US disclosed
US-7897964-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2011-03-01 US disclosed
US-7816668-B2 comprising carbazole rings, contained within hole transporting layer of light emitting element; high glass transistion temperature, heat resistance, and small power consumption SEMICONDUCTOR ENERGY LABORATORY CO., LTD 2010-10-19 US disclosed
US-20100244693-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2010-09-30 US disclosed
WO-2008105349-A1 LIGHT-EMITTING ELEMENT USING SPIROFLUORENE DERIVATIVE AND ELECTRONIC APPLIANCE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-09-04 WO disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
US-20070215867-A1 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2007-09-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 KDM4E 4076/4885ATM 833/4885L3MBTL1 1468/4885
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 KDM4E 4076/4885ATM 833/4885L3MBTL1 1468/4885
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 KDM4E 4076/4885ATM 833/4885L3MBTL1 1468/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.