SCHEMBL12560163

SCHEMBL12560163

Cc1ccc2c(c1)c1cc(C)ccc1n2-c1ccc(N(c2ccccc2)c2ccc3c(c2)C2(c4ccccc4-c4ccccc42)c2ccccc2-3)cc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.34
APP P05067 1/20 0.33
MAPT P10636 1/20 0.31
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
GAA P10253 1/20 0.30
GFER P55789 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13133854 0.97 KDM4E (0.35) PDK2APPBCHEACHE
SCHEMBL12560026 0.97 PDK2 (0.33) PDK2APPMAPTGAAGFER
SCHEMBL12560172 0.93 PDK2 (0.34) PDK2
SCHEMBL12560198 0.93 PDK2 (0.32) PDK2
SCHEMBL12560112 0.92 KDM4E (0.37) PDK2APP
SCHEMBL12559999 0.91 KDM4E (0.38) PDK2GAAGFER
SCHEMBL12362638 0.91 PDK2 (0.37) PDK2
SCHEMBL12704814 0.90 PGR (0.35) PDK2APPMAPT
SCHEMBL12560180 0.89
SCHEMBL12560185 0.89 PLA2G4A (0.33) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2018-06-21 US disclosed
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2018-06-21 US disclosed
US-9899602-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2018-02-20 US disclosed
US-9899602-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2018-02-20 US disclosed
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2017-05-04 US disclosed
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2017-05-04 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-9548457-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORIES CO., LTD. (JP) 2017-01-17 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LAB (JP) 2016-03-24 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
US-8304094-B2 High light efficincy; hole transporting substance; phosphorescence SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2012-11-06 US disclosed
US-20110147728-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2011-06-23 US disclosed
US-7897964-B2 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2011-03-01 US disclosed
US-7816668-B2 comprising carbazole rings, contained within hole transporting layer of light emitting element; high glass transistion temperature, heat resistance, and small power consumption SEMICONDUCTOR ENERGY LABORATORY CO., LTD 2010-10-19 US disclosed
US-20100244693-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2010-09-30 US disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
US-20080206598-A1 Light-emitting element using spirofluorene derivative and electronic appliance SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2008-08-28 US disclosed
US-20070215867-A1 Spirofluorene derivative, material for light-emitting element, light-emitting element, light-emitting device, and electronic device SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2007-09-20 US disclosed
WO-2007043354-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE SEMICONDUCTOR ENERGY LABORATORY CO., LTD. (JP) 2007-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170125679-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 PDK2 960/4885APP 3908/4885MAPT 4329/4885
US-20180175295-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 PDK2 960/4885APP 3908/4885MAPT 4329/4885
US-20160087209-A1 SPIROFLUORENE DERIVATIVE, MATERIAL FOR LIGHT-EMITTING ELEMENT, LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, AND ELECTRONIC DEVICE GRK1, PTGER2, PTGER1 PDK2 960/4885APP 3908/4885MAPT 4329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.