SCHEMBL1256802

SCHEMBL1256802

CCCCCc1ccc(O)c(N)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT8 Q9H7Z6 2/20 0.57
IGF1R P08069 2/20 0.53
ALOX15 P16050 2/20 0.53
ESR1 P03372 2/20 0.53
ADRA2A P08913 2/20 0.53
ADORA3 P0DMS8 2/20 0.53
TACR2 P21452 2/20 0.53
SLC6A2 P23975 2/20 0.53
SLC6A4 P31645 2/20 0.53
SLC6A3 Q01959 2/20 0.53
CYP3A4 P08684 2/20 0.53
PTGS2 P35354 2/20 0.53
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
SHBG P04278 1/20 0.53
TP53 P04637 1/20 0.53
HSPD1 P10809 1/20 0.53
ADRB3 P13945 1/20 0.53
HTR2C P28335 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9376917 0.98 KAT8 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL9001576 0.98 KAT8 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL9586309 0.98 KAT8 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL1315795 0.98 KAT8 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL8937894 0.98 KAT8 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL76664 0.94 SKP2 (0.59) KAT8IGF1RALOX15ESR1ADRA2A
SCHEMBL11004150 0.88 ALOX15 (0.61) KAT8IGF1RALOX15ADRA2ASLC6A2
SCHEMBL11004234 0.88 ALOX15 (0.61) KAT8IGF1RALOX15ADRA2ASLC6A2
SCHEMBL1023135 0.86 CNR1 (0.64) ALOX15ADRA2ASLC6A2SLC6A3CYP3A4
SCHEMBL272900 0.86 ALOX15 (0.58) IGF1RALOX15ADRA2ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3419966-B1 UV-ABSORBING VINYLIC MONOMERS AND USES THEREOF ALCON INC (CH) 2020-03-25 EP disclosed
US-7879520-B2 comprising binding resin (polystyrene) and charge control agent including azo-type iron complex salt; electrography; wear resistance; offset resistance ORIENT CHEMICAL INDUSTRIES, LTD. (JP) 2011-02-01 US disclosed
EP-1868038-B1 Toner for developing electrostatic image and image formation process using it ORIENT CHEMICAL IND (JP) 2010-06-02 EP disclosed
US-20070292779-A1 Toner for developing electrostatic image and image formation process using it ORIENT CHEMICAL INDUSTRIES, LTD. (JP) 2007-12-20 US disclosed
EP-1868038-A2 Toner for developing electrostatic image and image formation process using it Orient Chemical Industries, Ltd. (JP) 2007-12-19 EP disclosed
US-20070054899-A1 Aromatase inhibitor compounds and uses thereof PARALLEL WIRELESS, INC. 2007-03-08 US disclosed
EP-1678170-A1 USE OF A COMPOUND OF FORMULA (I) AS AN INHIBITOR OF AROMATASE FOR THERAPEUTIC PURPOSES AND COMPOUNDS OF FORMULA (1) THEREAS Yang Ji Chemical Company Ltd. (KR) 2006-07-12 EP disclosed
WO-2005033104-A1 USE OF A COMPOUND OF FORMULA (I) AS AN INHIBITOR OF AROMATASE FOR THERAPEUTIC PURPOSES AND COMPOUNDS OF FORMULA (1) THEREAS YANG JI CHEMICAL COMPANY, LTD (KR) 2005-04-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070054899-A1 Aromatase inhibitor compounds and uses thereof CYP19A1, CYP17A1, HSD17B11 KAT8 2356/4885IGF1R 539/4885ALOX15 205/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.