SCHEMBL12587724

SCHEMBL12587724

CBc1cc(N(C)C(=O)N(C)C)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.44
P2RX1 P51575 1/20 0.40
TACR2 P21452 4/20 0.34
TP53 P04637 1/20 0.33
CES2 O00748 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLQ O75417 2/20 0.32
MLYCD O95822 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
TACR3 P29371 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12435510 0.85 TACR1 (0.54) TACR1P2RX1TACR2TP53CES2
SCHEMBL12436257 0.80 TACR1 (0.46) TACR1P2RX1TP53CES2MAPT
SCHEMBL11006983 0.78 TACR1 (0.57) TACR1P2RX1TACR2CES2MAPT
SCHEMBL12436182 0.78 NOTUM (0.46) TACR1P2RX1TP53CES2POLQ
SCHEMBL12436222 0.78 P2RX1 (0.51) TACR1P2RX1TACR2TP53CES2
SCHEMBL13994392 0.72 CES2 (0.41) TACR1CES2MAPTRXRARXRB
SCHEMBL12435720 0.70 TACR1 (0.50) TACR1P2RX1CES2MAPTMLYCD
SCHEMBL15397669 0.70 TACR1 (0.59) TACR1P2RX1CES2MAPTPOLQ
SCHEMBL79186 0.68 TACR1 (0.50) TACR1P2RX1TP53CES2POLQ
SCHEMBL12435579 0.67 MLYCD (0.57) TACR1P2RX1CES2MAPTPOLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2336105-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME Takeda Pharmaceutical Company Limited (JP) 2011-06-22 EP disclosed