Phloretin

Phloretin

SCHEMBL1260339

O=C(C=CC1C=CC=CC1)c1ccccc1.O=C(CCc1ccc(O)cc1)c1c(O)cc(O)cc1O

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 10/20 0.51
SLC5A2 P31639 8/20 0.51
CYP19A1 P11511 4/20 0.51
MAPT P10636 3/20 0.51
SLC28A3 Q9HAS3 3/20 0.51
HPGD P15428 3/20 0.51
HSD17B10 Q99714 3/20 0.51
GAA P10253 2/20 0.51
NFKB1 P19838 2/20 0.51
NFKB2 Q00653 2/20 0.51
RELA Q04206 2/20 0.51
KDM4E B2RXH2 2/20 0.51
CYP3A4 P08684 2/20 0.51
THRB P10828 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
MEN1 O00255 1/20 0.51
SLC16A3 O15427 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2598846 0.84 GPR52 (0.43) HPGDCYP3A4CYP2C9CYP2C19MEN1
Phenol SCHEMBL28311351 0.80 KMT2A (0.44) CYP19A1MAPTHPGDHSD17B10GAA
SCHEMBL29561663 0.78 MAPT (0.42) MAPTHPGDNFKB1NFKB2RELA
SCHEMBL28251467 0.78 MAPT (0.42) MAPTHPGDNFKB1NFKB2RELA
SCHEMBL30573 0.78 MAPT (0.42) MAPTHPGDNFKB1NFKB2RELA
SCHEMBL11851207 0.77 MAPT (0.41) MAPTHPGDNFKB1NFKB2RELA
SCHEMBL22720628 0.77 MAPT (0.41) MAPTHPGDNFKB1NFKB2RELA
Bicarbonate SCHEMBL28901195 0.77 MAPT (0.41) MAPTHPGDNFKB1NFKB2RELA
SCHEMBL27540791 0.77 MAPT (0.41) MAPTHPGDNFKB1NFKB2RELA
Methane SCHEMBL28134892 0.77 MAPT (0.41) MAPTHPGDNFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150374652-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THEREOF PERIO SCIENCES, LLC 2015-12-31 US claimed
CN-118284402-A Cosmetic composition comprising a high amount of retinol 莱雅公司 2024-07-02 CN disclosed
CN-118201589-A Cosmetic composition comprising a high amount of ceramide-NP 莱雅公司 2024-06-14 CN disclosed
CN-118201586-A Cosmetic composition comprising a high amount of hydroxypropyl tetrahydropyran triol 莱雅公司 2024-06-14 CN disclosed
CN-117242185-A Biocatalytic preparation of dihydrochalcone 西姆莱斯有限公司 2023-12-15 CN disclosed
EP-4274430-A1 NOVEL COMPOSITIONS FOR SOUR TASTE BALANCING Symrise AG (DE) 2023-11-15 EP disclosed
CN-115996697-A Cosmetic composition with improved penetration 莱雅公司 2023-04-21 CN disclosed
WO-2022148540-A1 NOVEL COMPOSITIONS FOR SOUR TASTE BALANCING SYMRISE AG (DE) 2022-07-14 WO disclosed
EP-2370069-B1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THEREOF PERIO SCIENCES LLC (US) 2020-09-30 EP disclosed
WO-2016016826-A1 METHODS AND MATERIALS FOR MANIPULATING PHLORIDZIN PRODUCTION DARE ANDREW PATRICK (NZ) 2016-02-04 WO disclosed
EP-2235051-B1 GLYCOSYLTRANSFERASES, POLYNUCLEOTIDES ENCODING THESE AND METHODS OF USE NZ INST PLANT & FOOD RES LTD (NZ) 2015-09-30 EP disclosed
US-8859848-B2 Phloretin glycosyltransferases, polynucleotides encoding these and methods of use THE NEW ZEALAND INSTITUTE FOR PLANT AND FOOD RESEARCH LIMITED (NZ) 2014-10-14 US disclosed
US-20140050675-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THEREOF PERIO SCIENCES, LLC 2014-02-20 US disclosed
EP-2370069-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THERE Perio Sciences, LLC (US) 2011-10-05 EP disclosed
US-20110077275-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THEREOF PERIO SCIENCES, LLC 2011-03-31 US disclosed
US-20110030098-A1 Glycosyltransferases, Polynucleotides Encoding These And Methods Of Use THE NEW ZEALAND INSTITUTE FOR PLANT AND FOOD RESEARCH LIMITED (NZ) 2011-02-03 US disclosed
EP-2235051-A2 GLYCOSYLTRANSFERASES, POLYNUCLEOTIDES ENCODING THESE AND METHODS OF USE The New Zealand Institute for Plant and Food Research Limited (NZ) 2010-10-06 EP disclosed
US-20100183524-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THEREOF PERIO SCIENCES, LLC (US) 2010-07-22 US disclosed
WO-2010062835-A1 ANTIOXIDANT COMPOSITIONS FOR SOFT ORAL TISSUE AND METHODS OF FORMULATION AND USE THERE PERIO SCIENCES, LLC (US) 2010-06-03 WO disclosed
WO-2009082243-A2 GLYCOSYLTRANSFERASES, POLYNUCLEOTIDES ENCODING THESE AND METHODS OF USE THE NEW ZEALAND INSTITUTE FOR PLANT AND FOOD RESEARCH LIMITED (NZ) 2009-07-02 WO disclosed