SCHEMBL12631978

SCHEMBL12631978

Cc1ccc(S(=O)(=O)NC(CN(C)C)CC2(O)CCCCC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.41
CA9 Q16790 5/20 0.41
CA1 P00915 3/20 0.41
CA4 P22748 1/20 0.41
TSHR P16473 3/20 0.40
HTT P42858 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 3/20 0.40
CA12 O43570 3/20 0.40
MMP2 P08253 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CYP3A4 P08684 1/20 0.40
UTS2R Q9UKP6 1/20 0.40
CA7 P43166 2/20 0.39
POLB P06746 1/20 0.39
PLAU P00749 1/20 0.39
HPN P05981 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1864898 0.85 CA2 (0.43) CA2CA9CA1CA4TSHR
SCHEMBL1867581 0.84 TSHR (0.43) CA2CA9CA1CA4TSHR
SCHEMBL1863476 0.83 MMP13 (0.38) CA2CA9CA1CA4TSHR
SCHEMBL1863742 0.82 TSHR (0.42) CA2CA9CA1CA4TSHR
SCHEMBL1863963 0.81 HSD17B10 (0.35) CA2CA9CA1CA4TSHR
SCHEMBL27829347 0.80 CA9 (0.43) CA2CA9CA1CA4TSHR
SCHEMBL4869315 0.77 SLC1A3 (0.48) CA2CA9CA1CA4TSHR
SCHEMBL4869319 0.77 SLC1A3 (0.48) CA2CA9CA1CA4TSHR
SCHEMBL1867972 0.77 TSHR (0.39) CA2CA9CA1CA4TSHR
SCHEMBL1862267 0.76 MMP13 (0.39) CA2CA9CA1CA4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455521-B2 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. (US) 2013-06-04 US disclosed
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. 2011-05-05 US disclosed
US-7754737-B2 Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS, INC. (US) 2010-07-13 US disclosed
US-20090018103-A1 Diaminoalkane Aspartic Protease Inhibitors VITAE PHARMACEUTICAL, INC (US) 2009-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110105506-A1 Diaminoalkane aspartic protease inhibitors DNPEP, PEPD, ACE CA2 1046/4885CA9 1585/4885CA1 149/4885
US-20090018103-A1 Diaminoalkane Aspartic Protease Inhibitors DNPEP, PEPD, ACE CA2 1046/4885CA9 1585/4885CA1 149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.