SCHEMBL12632565

SCHEMBL12632565

C=C(C)OCCCCN1CCN(c2cccc(-c3ccc4c(c3)C(C)(C)CCC4(C)C)n2)CC1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
HTR1A P08908 3/20 0.41
HTR2A P28223 2/20 0.41
DRD3 P35462 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
HRH3 Q9Y5N1 5/20 0.39
MAOB P27338 6/20 0.38
KCNH2 Q12809 2/20 0.38
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
MAOA P21397 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014838 0.91 RARA (0.46) RARARARBHTR1AHTR2ADRD3
SCHEMBL2011986 0.88 RARA (0.47) RARARARBHTR1AHTR2ADRD3
SCHEMBL2013156 0.88 RARA (0.43) RARARARBHTR1AHTR2ADRD3
SCHEMBL2049463 0.88 HTR1A (0.44) RARARARBHTR1AHTR2ADRD3
SCHEMBL12633279 0.86 RARA (0.43) RARARARBHTR1AHTR2ADRD3
SCHEMBL12633167 0.86 RARA (0.47) RARARARBHTR1AHTR2ADRD3
SCHEMBL2053886 0.85 HRH3 (0.43) RARARARBHTR1AHTR2ADRD3
SCHEMBL2013985 0.85 RARA (0.46) RARARARBHTR1AHTR2ADRD3
SCHEMBL12632929 0.85 RARA (0.46) RARARARBHTR1AHTR2ADRD3
SCHEMBL2013393 0.85 RARA (0.46) RARARARBHTR1AHTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072791-A1 SPHINGOSINE KINASE INHIBITORS MERCK PATENT GMBH (DE) 2011-06-23 WO disclosed