SCHEMBL12633192

SCHEMBL12633192

CCCCOc1ccc(-c2ccc3c(c2)C(C)(C)CCC3(C)C)nc1N1CCN(CCCCCO)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARG P13631 4/20 0.44
RARB P10826 4/20 0.44
RARA P10276 3/20 0.44
PDE5A O76074 9/20 0.40
KCNH2 Q12809 1/20 0.37
CTSS P25774 2/20 0.36
CTSK P43235 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
RXRA P19793 1/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15241245 0.98 RARG (0.45) RARGRARBRARAPDE5AKCNH2
SCHEMBL2014293 0.94 RARG (0.44) RARGRARBRARAPDE5AKCNH2
SCHEMBL12632960 0.82 RARA (0.43) RARGRARBRARAPDE5AKCNH2
SCHEMBL12633230 0.82 RARB (0.39) RARGRARBRARAPDE5AKCNH2
SCHEMBL2016394 0.81 RARG (0.45) RARGRARBRARAPDE5ADRD2
SCHEMBL15241246 0.81 RARB (0.39) RARGRARBRARAPDE5AKCNH2
SCHEMBL2016809 0.79 ACHE (0.39) RARGRARBRARADRD2
SCHEMBL12633904 0.79 CKS1B (0.42) RARGRARBRARARXRA
SCHEMBL2015010 0.78 RARG (0.43) RARGRARBRARAPDE5ADRD2
SCHEMBL2012292 0.78 ACHE (0.40) RARGRARBRARADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072791-A1 SPHINGOSINE KINASE INHIBITORS MERCK PATENT GMBH (DE) 2011-06-23 WO disclosed