SCHEMBL12643104

SCHEMBL12643104

O=Cc1cn(CCOCCO)c2c(OC(F)(F)F)cccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
MAPT P10636 3/20 0.37
ALDH1A1 P00352 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR2 P34972 2/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
ERBB3 P21860 1/20 0.35
ERBB4 Q15303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12643055 0.90 TDP1 (0.39) TDP1MAPTALDH1A1NPC1RAB9A
SCHEMBL2040251 0.82 IDO1 (0.42) CNR2HTTLMNARORC
SCHEMBL2037470 0.82 ALDH1A1 (0.42) MAPTALDH1A1MEN1KMT2ACNR2
SCHEMBL12643061 0.81 CNR2 (0.43) TDP1MAPTALDH1A1NPC1RAB9A
SCHEMBL12642956 0.80 POLB (0.44) TDP1MAPTALDH1A1NPC1RAB9A
SCHEMBL2036078 0.75 EGFR (0.42) MAPTMEN1KMT2AEGFRERBB2
SCHEMBL16222983 0.73 POLB (0.60) TDP1MAPTALDH1A1NPC1RAB9A
SCHEMBL2036160 0.72 IDO1 (0.41) CNR2HTTLMNARORC
SCHEMBL2044112 0.71 HTT (0.46) CNR2HTTLMNARORC
SCHEMBL2036957 0.71 RORC (0.43) MAPTALDH1A1MEN1KMT2ACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079102-A1 INDOLYL-PIPERIDINYL BENZYLAMINES AS BETA-TRYPTASE INHIBITORS SANOFI (FR) 2011-06-30 WO disclosed