SCHEMBL12674686

SCHEMBL12674686

CCOC(=O)CN1C(=O)C(Cl)(Cl)c2cc(Br)ccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 2/20 0.48
ELANE P08246 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ANPEP P15144 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PKM P14618 1/20 0.45
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
ALDH3A1 P30838 2/20 0.44
ALDH2 P05091 1/20 0.44
HTT P42858 2/20 0.44
USP2 O75604 1/20 0.44
PIN1 Q13526 1/20 0.44
PIN4 Q9Y237 1/20 0.44
MAPT P10636 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5956251 0.81 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1LMNAELANE
SCHEMBL13224465 0.79 CYP1A2 (0.44) ALDH1A1KMT2AMEN1LMNAELANE
SCHEMBL12674685 0.74 ALDH1A1 (0.76) ALDH1A1KMT2ALMNAGSK3AGSK3B
SCHEMBL26640417 0.74 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1ANPEPSMN1; SMN2
SCHEMBL30642153 0.74 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1ANPEPSMN1; SMN2
SCHEMBL14876494 0.73 PTGDR2 (0.49) ALDH1A1KMT2AMEN1USP2
SCHEMBL15522229 0.72 HDAC1 (0.53) ALDH1A1KMT2AMEN1LMNACYP1A2
SCHEMBL522944 0.72 PIN1 (0.68) ALDH1A1KMT2AMEN1LMNAGSK3A
SCHEMBL7371898 0.71 ALDH1A1 (0.65) ALDH1A1LMNAELANESMN1; SMN2GSK3A
SCHEMBL6316299 0.71 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056985-A2 SUBSTITUTED HETEROCYCLIC COMPOUNDS GILEAD SCIENCES, INC. (US) 2011-05-12 WO disclosed