SCHEMBL12700552

SCHEMBL12700552

Cc1ccc(-n2cc(C=O)c3cc(F)ccc32)cc1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
KDM4E B2RXH2 3/20 0.61
KCNH2 Q12809 9/20 0.44
SCN2B O60939 1/20 0.40
SCN1A P35498 1/20 0.40
SCN1B Q07699 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
KAT2B Q92831 1/20 0.40
UBE2N P61088 1/20 0.39
RORC P51449 1/20 0.39
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8418393 0.81 ALDH1A1 (0.65) ALDH1A1KCNH2
SCHEMBL2134631 0.78 KDM4E (0.67) ALDH1A1KDM4EUBE2N
SCHEMBL3716522 0.77 ALDH1A1 (1.00) ALDH1A1KDM4EUBE2NKMT2A
SCHEMBL3972960 0.77 ALDH1A1 (0.59) ALDH1A1KDM4EKCNH2SCN2BSCN1A
SCHEMBL1092202 0.76 ALDH1A1 (1.00) ALDH1A1KDM4EKMT2A
SCHEMBL3233050 0.73 ALDH1A1 (0.66) ALDH1A1KDM4EKMT2A
SCHEMBL12182481 0.73 ALDH1A1 (0.65) ALDH1A1KDM4EKMT2A
SCHEMBL1093920 0.73 ALDH1A1 (0.65) ALDH1A1KDM4EKMT2A
SCHEMBL27431558 0.72 ALDH1A1 (0.63) ALDH1A1KDM4EKMT2A
SCHEMBL8238735 0.71 ALDH1A1 (0.66) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101487-A1 DI/TRI-AZA-SPIRO-C9-C11ALKANES NOVARTIS AG (CH) 2012-08-02 WO disclosed