SCHEMBL12719566

SCHEMBL12719566

COc1nc2ccccc2cc1NC(=O)Nc1cccc(Oc2ccnc(C(N)=O)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
RAF1 P04049 6/20 0.45
MAPT P10636 2/20 0.45
RET P07949 2/20 0.44
BRAF P15056 5/20 0.44
KDR P35968 3/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 1/20 0.43
GRM4 Q14833 1/20 0.43
CDK8 P49336 2/20 0.42
HTT P42858 1/20 0.42
PLK4 O00444 1/20 0.42
AURKA O14965 1/20 0.42
MAPK13 O15264 1/20 0.42
JAK2 O60674 1/20 0.42
MAP4K4 O95819 1/20 0.42
ABL1 P00519 1/20 0.42
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4173358 0.92 RAF1 (0.52) RAF1MAPTRETKDRPLK4
SCHEMBL4181174 0.90 RET (0.56) RAF1RETBRAFKDRCDK8
SCHEMBL257963 0.82 RAF1 (0.59) RAF1RETBRAFKDRCDK8
SCHEMBL938402 0.78 RAF1 (0.58) RAF1MAPTBRAFKDRALDH1A1
SCHEMBL261957 0.76 MAPT (0.49) RAB9ANPC1MAPTALDH1A1KDM4E
SCHEMBL1395927 0.76 RAF1 (0.68) RAF1RETBRAFKDRCDK8
SCHEMBL16990709 0.75 ALDH1A1 (0.46) RAB9ANPC1ALDH1A1KDM4EMEN1
SCHEMBL939310 0.74 ALDH1A1 (0.46) RAF1MAPTBRAFKDRALDH1A1
SCHEMBL4185779 0.74 RAF1 (0.58) RAB9ANPC1RAF1BRAFKDR
SCHEMBL12749714 0.74 MEN1 (0.47) RAF1KDRKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7928239-B2 Anticarcinogenic agents BAYER HEALTHCARE LLC (US) 2011-04-19 US disclosed
US-7928239-B2 Anticarcinogenic agents BAYER HEALTHCARE LLC (US) 2011-04-19 US disclosed