SCHEMBL12720437

SCHEMBL12720437

CC(=O)CNC(=O)C1=C(O)c2ccc(Cl)cc2C(C)(C)C1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.38
SPR P35270 2/20 0.38
EGLN1 Q9GZT9 4/20 0.37
IDO1 P14902 3/20 0.36
TDO2 P48775 1/20 0.36
PTGDR Q13258 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
VEGFA P15692 1/20 0.35
FLT1 P17948 1/20 0.35
POLB P06746 1/20 0.33
THRB P10828 1/20 0.33
RECQL P46063 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PSMB11 A5LHX3 1/20 0.33
PSMA7 O14818 1/20 0.33
NFKB1 P19838 1/20 0.33
PSMB1 P20618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12720376 0.91 SPR (0.44) CYP11B2SPREGLN1IDO1TDO2
SCHEMBL1626702 0.91 EGLN1 (0.46) SPREGLN1PTGDRPTGDR2VEGFA
SCHEMBL12720429 0.87 CYP11B2 (0.36) CYP11B2SPREGLN1IDO1TDO2
SCHEMBL12720433 0.86 SPR (0.38) SPREGLN1PSMB11PSMA7PSMB1
SCHEMBL12720448 0.86 SPR (0.38) SPREGLN1PTGDR2L3MBTL1PSMB11
SCHEMBL1627289 0.85 PTPRC (0.43) SPREGLN1IDO1PTGDRPTGDR2
SCHEMBL12720458 0.85 SPR (0.39) SPREGLN1
SCHEMBL12720503 0.85 SPR (0.44) SPREGLN1ALDH1A1POLBMEN1
SCHEMBL12720427 0.84 SPR (0.42) SPREGLN1IDO1TDO2
SCHEMBL12720435 0.83 SPR (0.36) SPREGLN1PTGDR2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7928139-B2 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof AMGEN INC. (US) 2011-04-19 US disclosed
US-20100048572-A1 NAPHTHALENONE COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF AMGEN INC. (US) 2010-02-25 US disclosed
US-7635715-B2 Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof AMGEN INC. (US) 2009-12-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048572-A1 NAPHTHALENONE COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF EGLN2, EGLN3, HIF1AN CYP11B2 44/4885SPR 754/4885EGLN1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.