SCHEMBL12721815

SCHEMBL12721815

Bc1cnc2[nH]nc(N)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.38
LRRK2 Q5S007 2/20 0.38
PI4KA P42356 1/20 0.38
XDH P47989 1/20 0.38
PI4K2B Q8TCG2 1/20 0.38
PI4K2A Q9BTU6 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
DYRK1A Q13627 2/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
JAK2 O60674 5/20 0.32
PDPK1 O15530 4/20 0.32
KDM4E B2RXH2 1/20 0.32
CYP3A4 P08684 1/20 0.32
GAA P10253 1/20 0.32
CHEK1 O14757 1/20 0.31
AURKA O14965 1/20 0.31
DAPK3 O43293 1/20 0.31
MAP4K4 O95819 1/20 0.31
PAK4 O96013 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11927605 0.78
SCHEMBL14044896 0.76 NOS3 (0.47) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL30440210 0.76 RET (0.38) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL12466822 0.76 IDO1 (0.46) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL175432 0.76 RET (0.38) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL1585071 0.76 DYRK1A (0.55) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL30508312 0.76 DYRK1A (0.55) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL12721812 0.74 CHEK1 (0.41) GSK3AGSK3BCHEK1AURKA
SCHEMBL7216007 0.73 RET (0.36) RETLRRK2PI4KAXDHPI4K2B
SCHEMBL12515294 0.73 HAO1 (0.37) GSK3AGSK3BPRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011044157-A1 HETEROCYCLIC COMPOUNDS USEFUL AS PDK1 INHIBITORS BIOGEN IDEC MA INC. (US) 2011-04-14 WO disclosed