SCHEMBL1272672

SCHEMBL1272672

COc1c(C)c(=O)[nH]c2nc(N(C)C)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.45
ADORA1 P30542 2/20 0.45
KDM4E B2RXH2 3/20 0.42
KMT2A Q03164 2/20 0.42
MAPK13 O15264 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
LMNA P02545 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
XBP1 P17861 1/20 0.34
HTT P42858 1/20 0.34
CLK1 P49759 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
TDP2 O95551 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11588963 0.79 ADORA1 (0.51) ADORA2AADORA1KDM4EKMT2AMAPK14
SCHEMBL3019661 0.72 ADORA2A (0.49) ADORA2AADORA1KDM4EKMT2AMAPK13
SCHEMBL11591825 0.61 KDM4E (0.58) ADORA2AADORA1KDM4EKMT2AALDH1A1
SCHEMBL5369123 0.61 KDM4E (0.50) ADORA2AADORA1KDM4EKMT2ALMNA
SCHEMBL11589180 0.61 ADORA1 (0.58) ADORA2AADORA1KDM4EKMT2AMAPK13
SCHEMBL22666569 0.60 ADORA2A (0.42) ADORA2AADORA1MAPK13MAPK12MAPK11
SCHEMBL3358664 0.60 AURKA (0.54) ADORA2AADORA1KDM4EKMT2AALDH1A1
SCHEMBL4529800 0.59 PDE3B (0.50) ADORA2AADORA1LMNAALDH1A1MAPT
SCHEMBL22666800 0.58 ADORA2A (0.40) ADORA2AADORA1MAPK13MAPK12MAPK11
SCHEMBL76177 0.58 KDM4E (0.56) ADORA1KDM4EALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016043983-A1 COMPOSITION WITH HIGH FILM FLEX ENDURANCE AND ARTICLES DERIVED THEREFROM SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2016-03-24 WO disclosed
WO-2014072923-A1 PROCESS FOR PRODUCING POLYCARBONATE COMPOSITIONS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-05-15 WO disclosed
WO-2014066784-A1 LIGHT EMITTING DIODE DEVICES, METHOD OF MANUFACTURE, USES THEREOF SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-05-01 WO disclosed
WO-2014053878-A1 SUSTAINABLE ISOSORBIDE - CONTAINING POLYCARBONATE - POLYLACTIDE BLENDS SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2014-04-10 WO disclosed
EP-2379640-A1 THERMOPLASTIC COMPOSITION WITH IMPROVED LOW TEMPERATURE DUCTILITY SABIC Innovative Plastics IP B.V. (NL) 2011-10-26 EP disclosed
WO-2011082054-A1 POLYCARBONATE-POLY(ETHER-ESTER) COPOLYMER COMPOSITION, METHOD OF MANUFACTURE, AND ARTICLES THEREFROM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2011-07-07 WO disclosed
WO-2011028511-A1 FLAME RETARDANT THERMOPLASTIC POLYCARBONATE COMPOSITIONS AND FILMS MADE THEREFROM SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2011-03-10 WO disclosed
EP-2291454-A1 POLYMER COMPOSITIONS, METHOD OF MANUFACTURE, AND ARTICLES FORMED THEREFROM SABIC Innovative Plastics IP B.V. (NL) 2011-03-09 EP disclosed
WO-2011014778-A1 FLAME-RETARDANT REINFORCED POLYCARBONATE COMPOSITIONS SABIC INNOVATIVE PLASTICS IP B.V (NL) 2011-02-03 WO disclosed
EP-2104698-A1 MONOMERS FOR THE PREPARATION OF SILYLATED POLYCARBONATE POLYMERS Momentive Performance Materials Inc. (US) 2009-09-30 EP disclosed
EP-1940958-A2 FLAME RETARDANT THERMOPLASTIC POLYCARBONATE COMPOSITIONS, METHOD OF MANUFACTURE, AND METHOD OF USE THEREOF GENERAL ELECTRIC COMPANY (a New York Corporation) (US) 2008-07-09 EP disclosed
WO-2008079358-A1 MONOMERS FOR THE PREPARATION OF SILYLATED POLYCARBONATE POLYMERS MOMENTIVE PERFORMANCE MATERIALS INC. (US) 2008-07-03 WO disclosed
EP-1856196-A1 PROTECTED POLYCARBONATE FILMS HAVING THERMAL AND UV RADIATION STABILITY, AND METHOD OF MAKING General Electric Company (US) 2007-11-21 EP disclosed
WO-2007081509-A2 POLYCARBONATE COMPOSITIONS AND ARTICLES FORMED THEREFROM, WITH MATTE SURFACES AND HIGH LIGHT TRANSMISSIONS GENERAL ELECTRIC COMPANY (US) 2007-07-19 WO disclosed
WO-2007070530-A2 THERMOPLASTIC POLYCARBONATE COMPOSITIONS, METHOD OF MANUFACTURE, AND METHOD OF USE THEREOF GENERAL ELECTRIC COMPANY (US) 2007-06-21 WO disclosed
WO-2007050412-A2 FLAME RETARDANT THERMOPLASTIC POLYCARBONATE COMPOSITIONS, METHOD OF MANUFACTURE, AND METHOD OF USE THEREOF GENERAL ELECTRIC COMPANY (US) 2007-05-03 WO disclosed
WO-2006088893-A1 PROTECTED POLYCARBONATE FILMS HAVING THERMAL AND UV RADIATION STABILITY, AND METHOD OF MAKING GENERAL ELECTRIC COMPANY (US) 2006-08-24 WO disclosed
EP-0126753-A4 STABILIZERS FOR DYE LASERS. UNIVERSITY PATENTS INC (US) 1986-11-05 EP disclosed
EP-0126753-A1 STABILIZERS FOR DYE LASERS UNIVERSITY PATENTS, INC. (US) 1984-12-05 EP disclosed
WO-1984001956-A1 STABILIZERS FOR DYE LASERS UNIVERSITY PATENTS INC (US) 1984-05-24 WO disclosed