SCHEMBL11588963

SCHEMBL11588963

COc1c(C)c(=O)[nH]c2nc(N)ccc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.51
ADORA2A P29274 2/20 0.51
KDM4E B2RXH2 3/20 0.44
KMT2A Q03164 2/20 0.44
CA5A P35218 1/20 0.41
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 2/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36
CLK1 P49759 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
XDH P47989 1/20 0.35
PARP1 P09874 1/20 0.35
MAPK14 Q16539 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11589180 0.82 ADORA1 (0.58) ADORA1ADORA2AKDM4EKMT2ACA5A
SCHEMBL1272672 0.79 ADORA2A (0.45) ADORA1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL11592378 0.71 ADORA1 (0.53) ADORA1ADORA2AKDM4EKMT2ACA5A
SCHEMBL8324129 0.70 ADORA1 (0.54) ADORA1ADORA2AKDM4EKMT2ACA5A
SCHEMBL7978388 0.68 ADORA1 (0.61) ADORA1ADORA2AKDM4EKMT2ACA5A
SCHEMBL5369123 0.66 KDM4E (0.50) ADORA1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL11591825 0.62 KDM4E (0.58) ADORA1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL14879331 0.61 ADORA1 (0.65) ADORA1ADORA2AKDM4ECA5ALMNA
SCHEMBL3358664 0.61 AURKA (0.54) ADORA1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL11591796 0.61 ADORA1 (0.53) ADORA1ADORA2AKDM4EKMT2ACA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4103257-A BLUE TO NEAR ULTRAVIOLET THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 1978-07-25 US disclosed